SCHEMBL10022673

SCHEMBL10022673

Cc1ccncc1-c1ncc(C(=O)O)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.49
CDC7 O00311 1/20 0.46
DBF4 Q9UBU7 1/20 0.46
ALDH1A1 P00352 3/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
SIRT3 Q9NTG7 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
DHODH Q02127 1/20 0.39
HPGD P15428 1/20 0.39
CYP1A2 P05177 3/20 0.38
CYP2E1 P05181 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C8 P10632 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2A6 P11509 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2B6 P20813 1/20 0.38
CYP2C19 P33261 1/20 0.38
ABL1 P00519 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27605419 0.87 CDC7 (0.45) CDC7DBF4ALDH1A1HDAC1HDAC6
SCHEMBL27817481 0.84 CDC7 (0.49) CDC7DBF4ALDH1A1HDAC1HDAC6
SCHEMBL28595774 0.83 CDC7 (0.69) CDC7DBF4ALDH1A1HDAC1HDAC6
SCHEMBL4283915 0.81 HPGD (0.55) HCAR2ALDH1A1HDAC1HDAC6HPGD
SCHEMBL10053508 0.77 CYP1A2 (0.44) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL12076008 0.77 HPGD (0.62) ALDH1A1TDP1HPGDCYP1A2CYP2E1
SCHEMBL22617526 0.76 SIRT3 (0.39) ALDH1A1SIRT3TDP1DHODHCYP1A2
SCHEMBL3593476 0.76 CDC7 (0.63) HCAR2CDC7DBF4ALDH1A1HDAC1
SCHEMBL24573406 0.73 HCAR2 (0.53) HCAR2CDC7DBF4ALDH1A1HDAC1
SCHEMBL6654343 0.73 ALDH1A1 (0.55) ALDH1A1HDAC6TDP1DHODHHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104642337-A Heterocyclic Compounds Used As Pesticides BAYER CROPSCIENCE AG 2015-05-27 CN disclosed
CN-102159079-B Heterocyclic compounds useful as pesticides BAYER CROPSCIENCE AG 2015-02-18 CN disclosed
EP-2590950-B1 N-CYCLYL-3-(CYCLYLCARBONYLAMINOMETHYL)BENZAMIDE DERIVATIVES AS RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2014-10-15 EP disclosed
US-20120165322-A1 RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-28 US disclosed
US-20120165322-A1 RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-28 US disclosed
CN-102159079-A Heterocyclic compounds useful as pesticides BAYER CROPSCIENCE AG 2011-08-17 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120165322-A1 RHO KINASE INHIBITORS ROCK1, ROCK2, RHOA HCAR2 2002/4885CDC7 567/4885DBF4 4324/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.