SCHEMBL10025823

SCHEMBL10025823

c1ccc2c(-n3c4ccc(cc4)c4ccccc4c4c5ccccc5c(c5ccccc5c5ccc(cc5)n(-c5cccc6ccccc56)c5ccccc53)c3ccccc34)cccc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.47
ALDH1A1 P00352 8/20 0.41
HSD17B10 Q99714 6/20 0.41
TSHR P16473 2/20 0.41
CYP2A6 P11509 1/20 0.41
CYP1A2 P05177 4/20 0.41
HPGD P15428 4/20 0.41
THRB P10828 1/20 0.41
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
HPRT1 P00492 1/20 0.39
POLB P06746 1/20 0.39
ERBB2 P04626 1/20 0.38
FYN P06241 1/20 0.38
MAOA P21397 1/20 0.38
ACHE P22303 1/20 0.38
AHR P35869 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10025810 0.79 KDM4E (0.50) TDP1ALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL17071084 0.77 TDP1 (0.45) TDP1ALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL17071128 0.76 TDP1 (0.44) TDP1ALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL490291 0.75 ALDH1A1 (0.50) TDP1ALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL29476055 0.75 ALDH1A1 (0.50) TDP1ALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL2627576 0.75 HSD17B10 (0.43) TDP1ALDH1A1HSD17B10TSHRCYP1A2
SCHEMBL14144351 0.75 TDP1 (0.46) TDP1ALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL14013692 0.74 TDP1 (0.44) TDP1ALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL23741500 0.74 TDP1 (0.41) TDP1ALDH1A1HSD17B10TSHRCYP1A2
Benzene SCHEMBL28312148 0.74 ALDH1A1 (0.53) TDP1ALDH1A1HSD17B10TSHRCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1859005-B1 NOVEL MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2016-04-27 EP disclosed
US-8124249-B2 Derivatives of fused aromatic systems; stability; sublimation stability; easy to purify due to better solubilty; easy reproducibility because do not form isomers MERCK PATENT GMBH (DE) 2012-02-28 US disclosed
US-8124249-B2 Derivatives of fused aromatic systems; stability; sublimation stability; easy to purify due to better solubilty; easy reproducibility because do not form isomers MERCK PATENT GMBH (DE) 2012-02-28 US disclosed
US-20080171225-A1 Novel Materials For Organic Electroluminescent Devices MERCK PATENT GMBH (DE) 2008-07-17 US disclosed
US-20080171225-A1 Novel Materials For Organic Electroluminescent Devices MERCK PATENT GMBH (DE) 2008-07-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080171225-A1 Novel Materials For Organic Electroluminescent Devices OR10J3, EML4, TYR TDP1 1990/4885ALDH1A1 1325/4885HSD17B10 3627/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.