SCHEMBL10028645

SCHEMBL10028645

O=C(c1cc(-c2ccncc2)cc(-c2cccnc2)c1)c1cc(-c2ccncc2)cc(-c2cccnc2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.57
MKNK1 Q9BUB5 7/20 0.56
MKNK2 Q9HBH9 7/20 0.56
ALDH1A1 P00352 2/20 0.50
CYP2A6 P11509 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP19A1 P11511 2/20 0.49
DYRK1A Q13627 2/20 0.45
EGFR P00533 1/20 0.45
FGFR1 P11362 1/20 0.45
KDR P35968 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL133437 0.93 KMO (0.64) KMOMKNK1MKNK2ALDH1A1CYP2A6
SCHEMBL12068188 0.86 CYP2A6 (0.68) MKNK1MKNK2ALDH1A1CYP2A6CYP1A2
SCHEMBL12070033 0.86 CYP2A6 (0.68) MKNK1MKNK2ALDH1A1CYP2A6CYP1A2
SCHEMBL133997 0.86 LMNA (0.50) ALDH1A1CYP1A2CYP3A4KDM4ELMNA
SCHEMBL24492814 0.82 CYP2A6 (0.62) KMOMKNK1MKNK2ALDH1A1CYP2A6
SCHEMBL17694301 0.82 CYP2A6 (0.62) KMOMKNK1MKNK2ALDH1A1CYP2A6
SCHEMBL22428552 0.82 CYP2A6 (0.62) KMOMKNK1MKNK2ALDH1A1CYP2A6
SCHEMBL22428539 0.82 CYP2A6 (0.62) KMOMKNK1MKNK2ALDH1A1CYP2A6
SCHEMBL16577179 0.82 CYP2A6 (0.62) KMOMKNK1MKNK2ALDH1A1CYP2A6
SCHEMBL27605046 0.81 KMO (0.77) KMOMKNK1MKNK2ALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9112172-B2 Organic electroluminescence device MERCK PATENT GMBH (DE) 2015-08-18 US disclosed
US-9112172-B2 Organic electroluminescence device MERCK PATENT GMBH (DE) 2015-08-18 US disclosed
US-20120037896-A1 ORGANIC ELECTROLUMINESCENCE DEVICE MERCK PATENT GMBH (DE) 2012-02-16 US disclosed
US-20120037896-A1 ORGANIC ELECTROLUMINESCENCE DEVICE MERCK PATENT GMBH (DE) 2012-02-16 US disclosed