Finafloxacin

Finafloxacin

SCHEMBL1002869

N#Cc1c(N2C[C@@H]3NCCO[C@H]3C2)c(F)cc2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

gyrAgyrBparCparE

The experimentally established mechanism targets of Finafloxacin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
KDM4E B2RXH2 4/20 0.54
HPGD P15428 4/20 0.54
HSD17B10 Q99714 3/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
KCNH2 Q12809 6/20 0.49
POLB P06746 2/20 0.49
OPRM1 P35372 2/20 0.49
PRKD3 O94806 1/20 0.49
ALOX15 P16050 1/20 0.49
CLK2 P49760 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
OPRD1 P41143 1/20 0.47
TOP2A P11388 5/20 0.43
TOP2B Q02880 5/20 0.43
LMNA P02545 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Finafloxacin SCHEMBL7608318 1.00 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDHSD17B10MEN1
Finafloxacin SCHEMBL7610665 1.00 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDHSD17B10MEN1
Finafloxacin SCHEMBL29378815 0.99 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDHSD17B10MEN1
Finafloxacin SCHEMBL7664508 0.99 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDHSD17B10MEN1
Finafloxacin SCHEMBL7660879 0.99 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL9182746 0.92 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL8803776 0.92 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL15791569 0.90 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7610667 0.90 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7608326 0.90 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 257 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12624057-B2 Bisphosphonate quinolone conjugates and uses thereof BIOVINC, LLC (US) 2026-05-12 US claimed
US-12329730-B2 Thermoresponsive hydrogel containing polymer microparticles for controlled drug delivery University of Pittsburgh—Of the Commonweatlh System of Higher Education (US) 2025-06-17 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-12312632-B2 Systems and methods for performing antimicrobial susceptibility testing SeLux Diagnostics, Inc. (US) 2025-05-27 US claimed
CN-118340907-A Polymer conjugates comprising bioactive agents 波利艾克蒂瓦有限公司 2024-07-16 CN claimed
US-20240182504-A1 BISPHOSPHONATE QUINOLONE CONJUGATES AND USES THEREOF BIOVINC LLC (US) 2024-06-06 US claimed
EP-3242667-B1 FINAFLOXACIN FOR USE IN THE TREATMENT OF URINARY TRACT INFECTIONS MERLION PHARMACEUTICALS GMBH (DE) 2024-06-05 EP claimed
US-11998615-B2 Functionalized nanoparticles and their use in treating bacterial infections THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2024-06-04 US claimed
US-20240102074-A1 SYSTEMS AND METHODS FOR PERFORMING ANTIMICROBIAL SUSCEPTIBILITY TESTING SeLux Diagnostics, Inc. 2024-03-28 US claimed
US-11845976-B2 Systems and methods for performing antimicrobial susceptibility testing SeLux Diagnostics, Inc. (US) 2023-12-19 US claimed
US-20220339293-A1 FUNCTIONALIZED NANOPARTICLES AND THEIR USE IN TREATING BACTERIAL INFECTIONS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2022-10-27 US claimed
US-11390900-B2 Antimicrobial cartridges and processes for multiplexed antimicrobial susceptibility testing SeLux Diagnostics, Inc. (US) 2022-07-19 US claimed
EP-4022079-A1 SYSTEMS AND METHODS FOR PERFORMING ANTIMICROBIAL SUSCEPTIBILITY TESTING Selux Diagnostics, Inc. (US) 2022-07-06 EP claimed
EP-3996751-A1 FUNCTIONALIZED NANOPARTICLES AND THEIR USE IN TREATING BACTERIAL INFECTIONS The Board Of Trustees Of The Leland Stanford Junior University (US) 2022-05-18 EP claimed
US-11291671-B2 Solid drug implants for intracochlear delivery of therapeutics for the treatment of Otic disorders O-RAY PHARMA, INC. (US) 2022-04-05 US claimed
WO-2022047234-A1 DRUG COMBINATION KITS AND METHODS OF DRUG DELIVERY PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2022-03-03 WO claimed
CN-105920603-B Treatment of erectile dysfunction and other indications 战略科学与技术有限责任公司 2022-02-11 CN claimed
WO-2022031761-A2 TARGETED DELIVERY OF THERAPEUTIC AGENTS SEPELO THERAPEUTICS, LLC (US) 2022-02-10 WO claimed
EP-0946176-B1 THE USE OF 7-(2-OXA-5,8-DIAZABICYCLO 4.3.0]NON-8-YL)-QUINOLONE CARBOXYLIC ACID AND NAPHTHYRIDON CARBOXYLIC ACID DERIVATIVES FOR MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF HELICOBACTER PYLORI INFECTIONS AND ASSOCIATED GASTRODUODENAL DISEASES BAYER AG (DE) 2002-03-27 EP claimed
US-6133260-A Use of 7-(2-oxa-5,8-diazabicyclo[4.3.0]non-8-yl)-quinolone carboxylic acid and naphthyridon carboxylic acid derivatives for the treatment of Helicobacter pylori infections and associated gastroduodenal diseases BAYER AKTIENGESELLSCHAFT (DE) 2000-10-17 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240182504-A1 BISPHOSPHONATE QUINOLONE CONJUGATES AND USES THEREOF BPGM, PHPT1, NQO2 ALDH1A1 2346/4885KDM4E 3437/4885HPGD 266/4885
US-12624057-B2 Bisphosphonate quinolone conjugates and uses thereof PTMS, CYP24A1, PHPT1 ALDH1A1 4057/4885KDM4E 476/4885HPGD 590/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.