SCHEMBL1002940

SCHEMBL1002940

CCSC(C)(Oc1ccc(F)c(F)c1F)C1CCCN1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.33
CYP2D6 P10635 3/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
CYP1A2 P05177 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C19 P33261 1/20 0.32
RAB9A P51151 1/20 0.32
HCRTR2 O43614 1/20 0.32
KCNH2 Q12809 1/20 0.31
HTR1A P08908 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HRH1 P35367 1/20 0.30
HTR2B P41595 1/20 0.30
SLC6A3 Q01959 1/20 0.30
TMEM97 Q5BJF2 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1002941 0.67 SLC6A2 (0.34) HCRTR2SLC6A3
SCHEMBL2044237 0.63 KDM4E (0.50) CYP2D6KDM4ENPC1CYP1A2HPGD
SCHEMBL7149465 0.63 CYP2D6 (0.34) CYP2D6HCRTR2KCNH2HTR1AHRH1
SCHEMBL24252041 0.62 HTR2C (0.34) HCRTR2KCNH2HTR2AHTR2CHTR2B
SCHEMBL10326466 0.61 CYP1A2 (0.41) TACR1CYP2D6KDM4ENPC1CYP1A2
SCHEMBL10326585 0.61 CYP1A2 (0.41) TACR1CYP2D6KDM4ENPC1CYP1A2
SCHEMBL10327169 0.61 CYP1A2 (0.41) TACR1CYP2D6KDM4ENPC1CYP1A2
SCHEMBL24252075 0.60 HTR2A (0.33) HTR2AHTR2CHTR2B
SCHEMBL17186941 0.59 ELANE (0.33) HTR2AHTR2CHTR2B
SCHEMBL13930842 0.59 KDM4E (0.35) CYP2D6KDM4ENPC1CYP1A2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011011231-A1 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS THERAVANCE, INC. (US) 2011-01-27 WO disclosed