SCHEMBL10033844

SCHEMBL10033844

NCCCNCCCCNCCCNC(=O)[C@H](N)CCCCNC(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.53
CNR1 P21554 3/20 0.51
CNR2 P34972 2/20 0.51
GRIN1 Q05586 2/20 0.50
GRIN2A Q12879 2/20 0.50
GNAI3 P08754 1/20 0.50
GNAO1 P09471 1/20 0.50
GNAI1 P63096 1/20 0.50
CHRNB2 P17787 3/20 0.48
CHRNB4 P30926 3/20 0.48
CHRNA3 P32297 3/20 0.48
CHRNA4 P43681 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12085454 1.00 MMP2 (0.53) MMP2CNR1CNR2GRIN1GRIN2A
SCHEMBL12085636 0.91 CNR1 (0.60) CNR1CNR2GRIN1GRIN2ACHRNB2
SCHEMBL10033846 0.85 GRIN1 (0.61) MMP2GRIN1GRIN2AGNAI3GNAO1
SCHEMBL12085474 0.85 GRIN1 (0.61) MMP2GRIN1GRIN2AGNAI3GNAO1
SCHEMBL20803506 0.84 CNR1 (0.69) CNR1CNR2
SCHEMBL12951413 0.83 HDAC3 (0.60) CNR1GRIN1GRIN2ACHRNB2CHRNB4
SCHEMBL24179776 0.83 GNAI3 (0.69) MMP2GRIN1GRIN2AGNAI3GNAO1
SCHEMBL12085475 0.83 GNAI3 (0.69) MMP2GRIN1GRIN2AGNAI3GNAO1
SCHEMBL10033848 0.83 GNAI3 (0.69) MMP2GRIN1GRIN2AGNAI3GNAO1
SCHEMBL17749476 0.83 CNR1 (0.67) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE43327-E1 Hydrophobic polyamine analogs and methods for their use AMINEX THERAPEUTICS, INC. (US) 2012-04-24 US disclosed
US-RE43327-E1 Hydrophobic polyamine analogs and methods for their use AMINEX THERAPEUTICS, INC. (US) 2012-04-24 US disclosed
US-7432302-B2 Composition containing polyamine transport inhibitor and use thereof MEDIQUEST THERAPEUTICS, INC. (US) 2008-10-07 US disclosed
US-7432302-B2 Composition containing polyamine transport inhibitor and use thereof MEDIQUEST THERAPEUTICS, INC. (US) 2008-10-07 US disclosed