SCHEMBL1003653

SCHEMBL1003653

C=C/C=C(\CCC)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 4/20 0.40
HDAC1 Q13547 4/20 0.40
HDAC2 Q92769 4/20 0.40
HDAC8 Q9BY41 4/20 0.40
FFAR3 O14843 3/20 0.40
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
TSHR P16473 5/20 0.33
GRIK1 P39086 3/20 0.32
GRIK2 Q13002 2/20 0.32
ALDH1A1 P00352 3/20 0.32
AKR1B1 P15121 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
BLM P54132 1/20 0.30
SLC6A3 Q01959 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17061403 1.00 HDAC3 (0.40) HDAC3HDAC1HDAC2HDAC8FFAR3
SCHEMBL1003654 1.00 HDAC3 (0.40) HDAC3HDAC1HDAC2HDAC8FFAR3
SCHEMBL8586760 0.87 CES1 (0.41) CES2CES1TSHRALDH1A1AKR1B1
SCHEMBL8586757 0.87 CES1 (0.41) CES2CES1TSHRALDH1A1AKR1B1
SCHEMBL28694016 0.85 AKR1B1 (0.46) CES2CES1TSHRALDH1A1AKR1B1
SCHEMBL31622773 0.84 GPR84 (0.48) CES2CES1TSHRALDH1A1AKR1B1
SCHEMBL19187723 0.83 TSHR (0.32) HDAC3HDAC1HDAC2HDAC8FFAR3
SCHEMBL4584135 0.81
SCHEMBL17265275 0.81
SCHEMBL6669152 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115812710-A Insect repellent composition comprising one or more insect repellent fatty acids having 9 to 21 carbon atoms 长荣置地有限公司 2023-03-21 CN disclosed
CN-112118739-B Insect repellent composition comprising one or more insect repellent fatty acids having 9 to 21 carbon atoms 长荣置地有限公司 2023-01-10 CN disclosed
US-11371063-B2 Microorganisms and methods for the production of butadiene using acetyl-coA GENOMATICA, INC. (US) 2022-06-28 US disclosed
CN-112118739-A Insect repellent composition comprising one or more insect repellent fatty acids having 9 to 21 carbon atoms 长荣置地有限公司 2020-12-22 CN disclosed
US-20200354753-A1 MICROORGANISMS AND METHODS FOR THE PRODUCTION OF BUTADIENE USING ACETYL-COA AGAIN BIO APS (DK) 2020-11-12 US disclosed
US-9463173-B2 Compositions and methods for treating obesity and obesity-related conditions THE JOHNS HOPKINS UNIVERSITY (US) 2016-10-11 US disclosed
US-20150250747-A1 COMPOSITIONS AND METHODS FOR TREATING OBESITY AND OBESITY-RELATED CONDITIONS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-09-10 US disclosed
EP-2694480-B1 ADAMANTYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2015-03-04 EP disclosed
EP-2456433-A2 METHODS FOR THE PREPARATION AND USE OF AQUEOUS SOLUTIONS OF MAGNESIUM VALPROATE HYDRATE AND L-CARNITINE Biolink Life Sciences, Inc. (US) 2012-05-30 EP disclosed
WO-2011011376-A2 METHODS FOR THE PREPARATION AND USE OF AQUEOUS SOLUTIONS OF MAGNESIUM VALPROATE HYDRATE AND L-CARNITINE BIOLINK LIFE SCIENCES, INC. (US) 2011-01-27 WO disclosed
US-20110015267-A1 METHODS FOR THE PREPARATION AND USE OF AQUEOUS SOLUTIONS OF MAGNESIUM VALPROATE HYDRATE AND L-CARNITINE BIOLINK LIFE SCIENCES, LLC 2011-01-20 US disclosed
US-20060223888-A1 Valproic acid analogues and pharmaceutical composition thereof THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2006-10-05 US disclosed
WO-2004054957-A2 VALPROIC ACID ANALOGUES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2004-07-01 WO disclosed
US-4432985-A N-alkylated carboxylic acid derivatives as anti-convulsant agents ABBOTT LABORATORIES (US) 1984-02-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060223888-A1 Valproic acid analogues and pharmaceutical composition thereof MALT1, HDAC11, GABRA6 HDAC3 8/4885HDAC1 5/4885HDAC2 14/4885
US-20110015267-A1 METHODS FOR THE PREPARATION AND USE OF AQUEOUS SOLUTIONS OF MAGNESIUM VALPROATE HYDRATE AND L-CARNITINE SLC25A20, CPT1A, CPT1B HDAC3 50/4885HDAC1 114/4885HDAC2 79/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.