SCHEMBL10036587

SCHEMBL10036587

Nc1ccc(C(c2ccc(N)c(C(O)(C(F)(F)F)C(F)(F)F)c2)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.54
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPK1 P28482 2/20 0.41
HSD17B10 Q99714 2/20 0.41
TSHR P16473 2/20 0.41
ALOX15 P16050 1/20 0.41
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
AR P10275 1/20 0.37
KIF11 P52732 2/20 0.35
GLA P06280 2/20 0.34
POLB P06746 2/20 0.34
GAA P10253 2/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12128592 0.93 SMN1; SMN2 (0.61) SMN1; SMN2MEN1KMT2AMAPK1HSD17B10
SCHEMBL7183547 0.85 KIF11 (0.42) SMN1; SMN2MAPK1TSHRESR1ESR2
SCHEMBL10002098 0.84 SMN1; SMN2 (0.41) SMN1; SMN2MEN1KMT2AMAPK1HSD17B10
SCHEMBL10036586 0.83 SMN1; SMN2 (0.57) SMN1; SMN2MEN1KMT2AMAPK1HSD17B10
SCHEMBL1635164 0.81 SMN1; SMN2 (0.67) SMN1; SMN2MEN1KMT2AMAPK1HSD17B10
SCHEMBL20869791 0.79 ESR1 (0.43) SMN1; SMN2MEN1KMT2AMAPK1HSD17B10
SCHEMBL18371620 0.79 SMN1; SMN2 (0.49) SMN1; SMN2MEN1KMT2AMAPK1HSD17B10
SCHEMBL10036673 0.78 SMN1; SMN2 (0.64) SMN1; SMN2MEN1KMT2AMAPK1HSD17B10
SCHEMBL6668409 0.77 FFAR4 (0.41) SMN1; SMN2HSD17B10TSHRESR1ESR2
SCHEMBL10002092 0.77 SMN1; SMN2 (0.45) SMN1; SMN2MEN1KMT2AMAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10384172-B2 Composite membrane with multi-layered active layer INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2019-08-20 US disclosed
US-10293308-B2 Antifouling and antimicrobial coatings for thin film composite membranes INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2019-05-21 US disclosed
US-20190015789-A1 ANTIFOULING AND ANTIMICROBIAL COATINGS FOR THIN FILM COMPOSITE MEMBRANES INTERNATIONAL BUSINESS MACHINES CORPORATION 2019-01-17 US disclosed
US-20170144113-A1 COMPOSITE MEMBRANE WITH MULTI-LAYERED ACTIVE LAYER INTERNATIONAL BUSINESS MACHINES CORPORATION 2017-05-25 US disclosed
US-9561474-B2 Composite membrane with multi-layered active layer INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2017-02-07 US disclosed
US-9504967-B2 Composite membrane with multi-layered active layer GLOBALFOUNDRIES INC. (KY) 2016-11-29 US disclosed
EP-2398840-B1 INTERFACIAL POLYMERIZATION METHODS FOR MAKING FLUOROALCOHOL-CONTAINING POLYAMIDES IBM (US) 2016-07-13 EP disclosed
US-20140353253-A1 COMPOSITE MEMBRANE WITH MULTI-LAYERED ACTIVE LAYER GLOBALFOUNDRIES U.S. INC. 2014-12-04 US disclosed
US-8857629-B2 Composite membrane with multi-layered active layer INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2014-10-14 US disclosed
US-8754139-B2 Polyamide membranes with fluoroalcohol functionality INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2014-06-17 US disclosed
US-8754139-B2 Polyamide membranes with fluoroalcohol functionality INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2014-06-17 US disclosed
US-20120012527-A1 COMPOSITE MEMBRANE WITH MULTI-LAYERED ACTIVE LAYER INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2012-01-19 US disclosed
US-20100216899-A1 POLYAMIDE MEMBRANES WITH FLUOROALCOHOL FUNCTIONALITY INTERNATIONAL BUSINESS MACHINES CORPORATION 2010-08-26 US disclosed
US-20100216899-A1 POLYAMIDE MEMBRANES WITH FLUOROALCOHOL FUNCTIONALITY INTERNATIONAL BUSINESS MACHINES CORPORATION 2010-08-26 US disclosed
WO-2010096563-A1 POLYAMIDE MEMBRANES WITH FLUOROALCOHOL FUNCTIONALITY INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2010-08-26 WO disclosed
WO-2010096565-A1 INTERFACIAL POLYMERIZATION METHODS FOR MAKING FLUOROALCOHOL-CONTAINING POLYAMIDES INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2010-08-26 WO disclosed
US-20100216967-A1 INTERFACIAL POLYMERIZATION METHODS FOR MAKING FLUOROALCOHOL-CONTAINING POLYAMIDES INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2010-08-26 US disclosed
US-20100216967-A1 INTERFACIAL POLYMERIZATION METHODS FOR MAKING FLUOROALCOHOL-CONTAINING POLYAMIDES INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2010-08-26 US disclosed