SCHEMBL1003723

SCHEMBL1003723

COC(=O)c1cc(C=O)c[nH]1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BAZ2B Q9UIF8 1/20 0.51
BAZ2A Q9UIF9 1/20 0.51
ALDH1A1 P00352 5/20 0.47
GAA P10253 2/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.41
CYP1A2 P05177 1/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
XDH P47989 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7497472 0.84 BAZ2B (0.50) BAZ2BBAZ2AALDH1A1GAALMNA
SCHEMBL23952005 0.82 BAZ2B (0.49) BAZ2BBAZ2AALDH1A1GAALMNA
SCHEMBL9197132 0.81 BAZ2B (0.47) BAZ2BBAZ2AALDH1A1GAALMNA
SCHEMBL261645 0.81 GABRP (0.47) BAZ2BBAZ2AALDH1A1GAALMNA
SCHEMBL4566308 0.80 BAZ2B (0.46) BAZ2BBAZ2AALDH1A1GAALMNA
SCHEMBL4566309 0.80 BAZ2B (0.46) BAZ2BBAZ2AALDH1A1GAALMNA
SCHEMBL19500071 0.80 TTR (0.47) BAZ2BBAZ2AALDH1A1GAALMNA
SCHEMBL27680446 0.78 NPC1 (0.54) BAZ2BBAZ2AALDH1A1GAALMNA
SCHEMBL643727 0.76 SMN1; SMN2 (0.43) ALDH1A1GAALMNAMAPK1
SCHEMBL28140695 0.76 MEN1 (0.46) BAZ2BBAZ2AALDH1A1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0434070-B1 Pyrrolealdehyde derivative MITSUBISHI CHEM CORP (JP) 1995-08-09 EP claimed
EP-0434070-A2 Pyrrolealdehyde derivative Mitsubishi Chemical Corporation (JP) 1991-06-26 EP claimed
CN-122055361-A Fascin inhibitors 北京双鹤润创科技有限公司 2026-05-15 CN disclosed
EP-4720054-A1 FASCIN INHIBITORS Beijing Double-Crane Runchuang Technology Co., Ltd. (CN) 2026-04-08 EP disclosed
US-12441724-B2 Inhibitors of plasma kallikrein and uses thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2025-10-14 US disclosed
WO-2025045233-A1 MACROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, AND USE THEREOF 劲方医药科技(上海)股份有限公司 2025-03-06 WO disclosed
EP-3930849-B1 THIAZOLE DERIVATIVES AS PROTEIN SECRETION INHIBITORS KEZAR LIFE SCIENCES (US) 2025-02-19 EP disclosed
WO-2024240245-A1 FASCIN INHIBITORS Beijing Double-Crane Runchuang Technology Co., Ltd. (CN) 2024-11-28 WO disclosed
US-20230078513-A1 INHIBITORS OF PLASMA KALLIKREIN AND USES THEREOF SHIRE HUMAN GENETIC THERAPIES, INC. 2023-03-16 US disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11352356-B2 Inhibitors of plasma kallikrein and uses thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2022-06-07 US disclosed
US-6066639-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2000-05-23 US disclosed
EP-0904271-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1999-03-31 EP disclosed
WO-1997041115-A1 5,6,7,8-TETRAHYDROPYRIDO[2,3-d]PYRIMIDINES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1997-11-06 WO disclosed
US-RE35096-E Antilipemic, anticholesterol, arteriosclerosis MITSUBISHI CHEMICAL CORPORATION (JP) 1995-11-21 US disclosed
EP-0434070-B1 Pyrrolealdehyde derivative MITSUBISHI CHEM CORP (JP) 1995-08-09 EP disclosed
US-5153217-A Antiiipemic, anticholesterol agents MITSUBISHI KASEI CORPORATION (JP) 1992-10-06 US disclosed
US-5082856-A Hyperlipemia, arteriosclerosis MITSUBISHI KASEI CORPORATION (JP) 1992-01-21 US disclosed
EP-0434070-A2 Pyrrolealdehyde derivative Mitsubishi Chemical Corporation (JP) 1991-06-26 EP disclosed
EP-0347902-A2 Pyrrolecarboxylic acid derivatives Mitsubishi Chemical Corporation (JP) 1989-12-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11352356-B2 Inhibitors of plasma kallikrein and uses thereof KLKB1, KLK1, KLK5 BAZ2B 1391/4885BAZ2A 1632/4885ALDH1A1 3157/4885
US-12441724-B2 Inhibitors of plasma kallikrein and uses thereof KLKB1, KLK1, KLK5 BAZ2B 1391/4885BAZ2A 1632/4885ALDH1A1 3157/4885
US-20230078513-A1 INHIBITORS OF PLASMA KALLIKREIN AND USES THEREOF KLKB1, KLK1, KLK5 BAZ2B 1391/4885BAZ2A 1632/4885ALDH1A1 3157/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.