SCHEMBL10037540

SCHEMBL10037540

Oc1ccc(-c2ccc(C3CCC(I)CC3)cc2)c(F)c1F

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 12/20 0.36
ESR1 P03372 6/20 0.36
CYP3A4 P08684 5/20 0.36
CYP2C9 P11712 4/20 0.36
APP P05067 2/20 0.34
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
QDPR P09417 1/20 0.32
FFAR4 Q5NUL3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25930081 0.86 CYP3A4 (0.45) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL25984723 0.85 ESR2 (0.36) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL14230677 0.85 ESR2 (0.53) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL15681401 0.84 CYP3A4 (0.47) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL15725311 0.82 CYP2C9 (0.49) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL3275306 0.81 ESR2 (0.43) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL3275302 0.81 ESR2 (0.43) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL10017626 0.81 ESR2 (0.33) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL15681399 0.79 HDAC2 (0.36) ESR2ESR1CYP3A4CYP2C9APP
SCHEMBL24221347 0.78 PDE4A (0.32) CYP3A4CYP2C9APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8168081-B2 Liquid-crystalline medium MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2012-05-01 US disclosed
US-20090309066-A1 Mixture of polar compounds containing cyclohexane and benzene rings some of which are vinylene-linked, especially containing fluoroalkoxy groups; for electrooptical twisted nematic monitor applications MERCK PATENT GESELLSCHAFT (DE) 2009-12-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090309066-A1 Mixture of polar compounds containing cyclohexane and benzene rings some of which are vinylene-linked, especially containing fluoroalkoxy groups; for electrooptical twisted nematic monitor applications VIM, CDH1, LEF1 ESR2 1692/4885ESR1 1399/4885CYP3A4 3869/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.