SCHEMBL10038523

SCHEMBL10038523

c1cc(-c2cccc3c2oc2ccc(-n4c5ccccc5c5ccccc54)cc23)cc(-c2cccc3c2oc2ccc(-n4c5ccccc5c5ccccc54)cc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.47
GGPS1 O95749 1/20 0.40
PRKDC P78527 11/20 0.38
PTGES2 Q9H7Z7 1/20 0.38
KDM4E B2RXH2 3/20 0.38
ATM Q13315 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
ALDH1A1 P00352 3/20 0.33
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
BRD4 O60885 2/20 0.33
BRD2 P25440 2/20 0.33
BRD3 Q15059 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
PDE2A O00408 1/20 0.33
PIK3C2A O00443 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17228745 0.96 ALOX5 (0.44) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL5029698 0.96 ALOX5 (0.46) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL17057192 0.95 ALOX5 (0.46) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL23505132 0.95 ALOX5 (0.44) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL5028289 0.93 ALOX5 (0.41) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL14733733 0.93 ALOX5 (0.44) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL5028179 0.93 ALOX5 (0.47) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL16573892 0.93 ALOX5 (0.50) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL18265970 0.92 ALOX5 (0.43) ALOX5GGPS1PRKDCPTGES2KDM4E
SCHEMBL20097818 0.92 ALOX5 (0.43) ALOX5GGPS1PRKDCPTGES2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10347850-B2 Organic electroluminescent element, lighting device and display device Konica Minolta, Inc. (JP) 2019-07-09 US disclosed
US-10177322-B2 Iridium complex, method for producing iridium complex, organic electroluminescent element, display device, and lighting device Konica Minolta, Inc. (JP) 2019-01-08 US disclosed
US-20170309839-A1 IRIDIUM COMPLEX, METHOD FOR PRODUCING IRIDIUM COMPLEX, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE KONICA MINOLTA INC (JP) 2017-10-26 US disclosed
US-20170309839-A1 IRIDIUM COMPLEX, METHOD FOR PRODUCING IRIDIUM COMPLEX, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE KONICA MINOLTA INC (JP) 2017-10-26 US disclosed
US-9748501-B2 Iridium complex, method for producing iridium complex, organic electroluminescent element, display device, and lighting device Konica Minolta, Inc. (JP) 2017-08-29 US disclosed
US-9748501-B2 Iridium complex, method for producing iridium complex, organic electroluminescent element, display device, and lighting device Konica Minolta, Inc. (JP) 2017-08-29 US disclosed
US-9673405-B2 Organic electroluminescent device, display apparatus, and lighting apparatus KONICA MINOLTA HOLDINGS, INC. (JP) 2017-06-06 US disclosed
US-9673405-B2 Organic electroluminescent device, display apparatus, and lighting apparatus KONICA MINOLTA HOLDINGS, INC. (JP) 2017-06-06 US disclosed
US-20160226006-A1 IRIDIUM COMPLEX, METHOD FOR PRODUCING IRIDIUM COMPLEX, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE Konica Minolta, Inc. (JP) 2016-08-04 US disclosed
US-20160226006-A1 IRIDIUM COMPLEX, METHOD FOR PRODUCING IRIDIUM COMPLEX, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE Konica Minolta, Inc. (JP) 2016-08-04 US disclosed
US-20130200340-A1 IRIDIUM COMPLEX COMPOUND, ORGANIC ELECTROLUMINESCENT ELEMENT MATERIAL, ORGANIC ELECTROLUMINESCENT ELEMENT, ILLUMINATION DEVICE AND DISPLAY DEVICE KONICA MINOLTA ADVANCED LAYERS, INC. (JP) 2013-08-08 US disclosed
US-20130119360-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, NEW COMPOUND FOR THE SAME, DISPLAY DEVICE AND LIGHTING DEVICE USING THE SAME MERCK PATENT GMBH (DE) 2013-05-16 US disclosed
US-20130099216-A1 ORGANIC ELECTROLUMINESCENT MATERIAL, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE AND LIGHTING DEVICE KONICA MINOLTA HOLDINGS, INC. (JP) 2013-04-25 US disclosed
US-20130099216-A1 ORGANIC ELECTROLUMINESCENT MATERIAL, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE AND LIGHTING DEVICE KONICA MINOLTA HOLDINGS, INC. (JP) 2013-04-25 US disclosed
EP-2584019-A1 ORGANIC ELECTROLUMINESCENT MATERIAL, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE AND LIGHTING DEVICE Konica Minolta Holdings, Inc. (JP) 2013-04-24 EP disclosed
US-8367224-B2 Organic electroluminescence element, new compound for the same, display device and lighting device using the same KONICA MINOLTA HOLDINGS, INC. (JP) 2013-02-05 US disclosed
US-20120018714-A1 ORGANIC ELECTROLUMINESCENT DEVICE, DISPLAY APPARATUS, AND LIGHTING APPARATUS KONICA MINOLTA HOLDINGS, INC. (JP) 2012-01-26 US disclosed
US-20120018714-A1 ORGANIC ELECTROLUMINESCENT DEVICE, DISPLAY APPARATUS, AND LIGHTING APPARATUS KONICA MINOLTA HOLDINGS, INC. (JP) 2012-01-26 US disclosed
US-20110006670-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, NEW COMPOUND FOR THE SAME, DISPLAY DEVICE AND LIGHTING DEVICE USING THE SAME KONICA MINOLTA HOLDINGS, INC. (JP) 2011-01-13 US disclosed
US-20110006670-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, NEW COMPOUND FOR THE SAME, DISPLAY DEVICE AND LIGHTING DEVICE USING THE SAME KONICA MINOLTA HOLDINGS, INC. (JP) 2011-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130200340-A1 IRIDIUM COMPLEX COMPOUND, ORGANIC ELECTROLUMINESCENT ELEMENT MATERIAL, ORGANIC ELECTROLUMINESCENT ELEMENT, ILLUMINATION DEVICE AND DISPLAY DEVICE INTS9, OCIAD1, INTS6 ALOX5 2532/4885GGPS1 1279/4885PRKDC 3896/4885
US-10177322-B2 Iridium complex, method for producing iridium complex, organic electroluminescent element, display device, and lighting device EED, SNW1, AP2M1 ALOX5 1708/4885GGPS1 2702/4885PRKDC 2772/4885
US-20170309839-A1 IRIDIUM COMPLEX, METHOD FOR PRODUCING IRIDIUM COMPLEX, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE EED, SNW1, AP2M1 ALOX5 1708/4885GGPS1 2702/4885PRKDC 2772/4885
US-20160226006-A1 IRIDIUM COMPLEX, METHOD FOR PRODUCING IRIDIUM COMPLEX, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE EED, SNW1, AP2M1 ALOX5 1708/4885GGPS1 2702/4885PRKDC 2772/4885
US-20110006670-A1 ORGANIC ELECTROLUMINESCENCE ELEMENT, NEW COMPOUND FOR THE SAME, DISPLAY DEVICE AND LIGHTING DEVICE USING THE SAME AOC2, AOC3, CDYL ALOX5 855/4885GGPS1 2906/4885PRKDC 3081/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.