SCHEMBL10039743

SCHEMBL10039743

c1ccc(CNC2CC3CNCC3C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.50
MC4R P32245 1/20 0.47
BCHE P06276 2/20 0.46
ACHE P22303 2/20 0.46
BACE1 P56817 2/20 0.46
FYN P06241 1/20 0.46
MEN1 O00255 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
KDM1A O60341 1/20 0.46
MAOA P21397 1/20 0.46
DPP8 Q6V1X1 2/20 0.44
DPP9 Q86TI2 2/20 0.44
DPP7 Q9UHL4 2/20 0.44
RB1 P06400 1/20 0.43
HRH2 P25021 1/20 0.42
ADRA1B P35368 1/20 0.42
OPRK1 P41145 1/20 0.42
SLC6A3 Q01959 1/20 0.42
OPRM1 P35372 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12323279 0.89 GRIN2B (0.47) GRIN2BBCHEACHEBACE1FYN
SCHEMBL8186106 0.85 GRIN2B (0.56) GRIN2BMC4RBCHEACHEBACE1
SCHEMBL4574649 0.81 CARM1 (0.50) CARM1PRMT6
SCHEMBL23948575 0.79 GRIN2B (0.50) GRIN2BBCHEACHEBACE1FYN
SCHEMBL14504603 0.78 GRIN2B (0.46) GRIN2BMC4RBCHEACHEBACE1
SCHEMBL28159653 0.78 GRIN2B (0.46) GRIN2BMC4RBCHEACHEBACE1
SCHEMBL28404369 0.78 GRIN2B (0.46) GRIN2BMC4RBCHEACHEBACE1
SCHEMBL7521305 0.77 GRIN2B (0.49) GRIN2BBCHEACHEBACE1FYN
SCHEMBL7161614 0.77 GRIN2B (0.49) GRIN2BBCHEACHEBACE1FYN
SCHEMBL6844239 0.77 GRIN2B (0.49) GRIN2BBCHEACHEBACE1FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012019430-A1 PHTHALAZINONE DERIVATIVE, AND PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-02-16 WO disclosed