SCHEMBL1004190

SCHEMBL1004190

COc1ccnc(CO)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.42
TLR8 Q9NR97 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
CYP2C9 P11712 3/20 0.40
ALDH1A1 P00352 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
DYRK1A Q13627 1/20 0.39
ATP4A P20648 3/20 0.38
ATP4B P51164 3/20 0.38
TSHR P16473 2/20 0.38
FYN P06241 1/20 0.37
CYP3A4 P08684 3/20 0.37
LMNA P02545 2/20 0.37
CYP1A2 P05177 2/20 0.37
ALOX15 P16050 2/20 0.37
PDE2A O00408 1/20 0.37
ABCC4 O15439 1/20 0.37
USP2 O75604 1/20 0.37
PDE5A O76074 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30963126 1.00 RAB9A (0.42) RAB9ATLR8TLR7CYP2C9ALDH1A1
Hydrochloric Acid SCHEMBL3181001 0.98 RAB9A (0.44) RAB9ATLR8TLR7CYP2C9ALDH1A1
SCHEMBL3186943 0.89 TLR8 (0.36) RAB9ATLR8TLR7CYP2C9ALDH1A1
SCHEMBL27863553 0.87 SMN1; SMN2 (0.43) RAB9ATLR8TLR7CYP2C9ALDH1A1
SCHEMBL3177121 0.85 DYRK1A (0.35) RAB9ATLR8TLR7CYP2C9ALDH1A1
SCHEMBL11918960 0.84 RAB9A (0.42) RAB9ATLR8TLR7CYP2C9ALDH1A1
SCHEMBL9079044 0.82 RAB9A (0.41) RAB9ATLR8TLR7CYP2C9ALDH1A1
SCHEMBL17434630 0.82 RAB9A (0.41) RAB9ATLR8TLR7CYP2C9ALDH1A1
SCHEMBL29446629 0.82 RAB9A (0.41) RAB9ATLR8TLR7CYP2C9ALDH1A1
SCHEMBL29694096 0.82 RAB9A (0.41) RAB9ATLR8TLR7CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 87 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109354587-A The preparation method and Pantoprazole Sodium of Pantoprazole Sodium 成都天台山制药有限公司 2019-02-19 CN claimed
CN-104557692-B A kind of preparation method of pantoprazole intermediate 2- chloromethyls -3,4- dimethoxy pyridine hydrochlorides 寿光富康制药有限公司 2018-08-21 CN claimed
CN-108191745-A The preparation method of 2- methylol -3,4- dimethoxy-pyridines 滁州学院 2018-06-22 CN claimed
CN-107011252-B The method for drawing azole intermediate and drug is prepared using the green technology for substituting the poisonous and harmful substances such as phosgene, thionyl chloride 浙江工业大学 2018-06-08 CN claimed
CN-107011252-A The method for drawing azole intermediate and medicine is prepared using the green technology for substituting the poisonous and harmful substances such as phosgene, thionyl chloride 浙江工业大学 2017-08-04 CN claimed
CN-104557692-A Preparation method of pantoprazole intermediate 2-chloromethyl-3,4-dimethoxy pyridine hydrochloride Shouguang fukang pharmaceutical co ltd 2015-04-29 CN claimed
CN-101875629-A Industrial preparation method of pantoprazole intermediate pyridine hydrochloride NANJING YUANHUA TECHNOLOGY CONSULTATION CO LTD 2010-11-03 CN claimed
WO-2025085492-A1 BORANE REDUCING REAGENTS EXACT SCIENCES CORPORATION (US) 2025-04-24 WO disclosed
CN-118324772-A Synthesis method and intermediate of furan [3,2-b ] pyridine derivative 北京颖诺凯胜科技有限公司 2024-07-12 CN disclosed
CN-115819403-A Preparation method of pantoprazole sodium 安徽普利药业有限公司 2023-03-21 CN disclosed
US-11241013-B2 Benzimidazole compounds as agricultural chemicals REDAG CROP PROT LTD (GB) 2022-02-08 US disclosed
US-11224224-B2 Thiobenzoimidazole as fungicides REDAG CROP PROTECTION LTD. (GB) 2022-01-18 US disclosed
US-20210204547-A1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS REDAG CROP PROT LTD (GB) 2021-07-08 US disclosed
US-4185103-A ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-01-22 US disclosed
EP-0004793-A2 2-nitro aminopyrimidone derivatives, a process for their preparation and their use to prepare 2-aminopyrimidone derivatives which have histamine H2-antagonist activity SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-10-17 EP disclosed
US-4159329-A BLOCKING AGENTS, ANTAGONISTS, ANTIHISTAMINES SMITHKLINE & FRENCH LABORATORIES LIMITED (GB) 1979-06-26 US disclosed
US-4156727-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-05-29 US disclosed
US-4154838-A ANTIHISTAMINE SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-05-15 US disclosed
US-4154834-A HETEROCYCLIC-(THIO)ALKYLAMINO SUBSTITUTED-4-PYRIMIDONE OR -THIONES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-05-15 US disclosed
US-4145546-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11224224-B2 Thiobenzoimidazole as fungicides CYP1B1, CYP51A1, CYP1A2 RAB9A 3497/4885TLR8 4016/4885TLR7 3996/4885
US-11241013-B2 Benzimidazole compounds as agricultural chemicals CYP3A4, CYP2C8, CYP2E1 RAB9A 4057/4885TLR8 3942/4885TLR7 4779/4885
US-20210204547-A1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS CYP3A4, CYP2C8, CYP2E1 RAB9A 4057/4885TLR8 3942/4885TLR7 4779/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.