SCHEMBL10042449

SCHEMBL10042449

c1ccc(-c2ccc3c(c2)c2cc(-c4ccc5[nH]c6ccccc6c5c4)ccc2n3-c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
AHR P35869 1/20 0.44
ATM Q13315 1/20 0.44
KIF11 P52732 3/20 0.43
PDE7A Q13946 2/20 0.42
PDE7B Q9NP56 2/20 0.42
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
GPR3 P46089 1/20 0.41
HPGD P15428 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 2/20 0.39
JAK2 O60674 1/20 0.39
LMNA P02545 1/20 0.38
GABRA1 P14867 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL263482 0.97 AHR (0.44) KDM4EL3MBTL1AHRATMKIF11
SCHEMBL25211466 0.97 AHR (0.44) KDM4EL3MBTL1AHRATMKIF11
SCHEMBL263499 0.97 AHR (0.44) KDM4EL3MBTL1AHRATMKIF11
SCHEMBL22198425 0.96 KDM4E (0.41) KDM4EL3MBTL1AHRATMKIF11
SCHEMBL15197844 0.96 KDM4E (0.51) KDM4EL3MBTL1AHRATMKIF11
SCHEMBL11998324 0.95 CDK4 (0.44) KDM4EL3MBTL1ATMPDE7APDE7B
SCHEMBL17234274 0.95 KDM4E (0.44) KDM4EL3MBTL1AHRATMKIF11
SCHEMBL17948128 0.95 KDM4E (0.44) KDM4EL3MBTL1AHRATMKIF11
SCHEMBL263170 0.94 AHR (0.42) KDM4EL3MBTL1AHRATMKIF11
SCHEMBL24228800 0.94 KDM4E (0.46) KDM4EL3MBTL1AHRATMKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12063855-B2 Compound for organic electric element, organic electric element using the same, and electronic device therefor DUK SAN NEOLUX CO., LTD. (KR) 2024-08-13 US disclosed
EP-4236652-A2 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES Merck Patent GmbH (DE) 2023-08-30 EP disclosed
EP-3328825-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2023-06-28 EP disclosed
US-11538995-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2022-12-27 US disclosed
US-20220367818-A1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT USING THE SAME, AND ELECTRONIC DEVICE THEREFOR DUK SAN NEOLUX CO., LTD. (KR) 2022-11-17 US disclosed
US-11322695-B2 Ink composition for organic light-emitting device, organic light-emitting device including film formed by using the ink composition, and method of manufacturing the organic light-emitting device SAMSUNG ELECTRONICS CO., LTD. (KR) 2022-05-03 US disclosed
EP-3577101-B1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2021-03-03 EP disclosed
EP-3712229-A1 MATERIALS FOR ELECTRONIC DEVICES Merck Patent GmbH (DE) 2020-09-23 EP disclosed
US-20200295273-A1 INK COMPOSITION FOR ORGANIC LIGHT-EMITTING DEVICE, ORGANIC LIGHT-EMITTING DEVICE INCLUDING FILM FORMED BY USING THE INK COMPOSITION, AND METHOD OF MANUFACTURING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO., LTD. (KR) 2020-09-17 US disclosed
EP-3027708-B1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2020-05-13 EP disclosed
WO-2014061991-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE CONTAINING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2014-04-24 WO disclosed
US-20140107338-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME Rohm, and Haas Electronic Materials Korea Ltd. (KR) 2014-04-17 US disclosed
US-20140107338-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME Rohm, and Haas Electronic Materials Korea Ltd. (KR) 2014-04-17 US disclosed
US-20140084271-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2014-03-27 US disclosed
US-20140084271-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2014-03-27 US disclosed
WO-2013085243-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-06-13 WO disclosed
WO-2013081416-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-06-06 WO disclosed
WO-2013073896-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-05-23 WO disclosed
WO-2013073874-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND AN ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-05-23 WO disclosed
WO-2012087007-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2012-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11538995-B2 Materials for organic electroluminescent devices L1CAM, EFNA1, EPCAM KDM4E 3061/4885L3MBTL1 2186/4885AHR 3734/4885
US-20140107338-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME OR10J3, VDAC2, KCNN2 KDM4E 826/4885L3MBTL1 910/4885AHR 3160/4885
US-11322695-B2 Ink composition for organic light-emitting device, organic light-emitting device including film formed by using the ink composition, and method of manufacturing the organic light-emitting device TYR, IK, TH KDM4E 137/4885L3MBTL1 108/4885AHR 163/4885
US-20200295273-A1 INK COMPOSITION FOR ORGANIC LIGHT-EMITTING DEVICE, ORGANIC LIGHT-EMITTING DEVICE INCLUDING FILM FORMED BY USING THE INK COMPOSITION, AND METHOD OF MANUFACTURING THE ORGANIC LIGHT-EMITTING DEVICE TYR, IK, TH KDM4E 137/4885L3MBTL1 108/4885AHR 163/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.