SCHEMBL10044941

SCHEMBL10044941

COc1cc(OC(F)F)cc(C)c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.42
POLB P06746 2/20 0.42
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 2/20 0.36
CYP3A4 P08684 1/20 0.36
CA9 Q16790 1/20 0.36
PDE2A O00408 2/20 0.36
PDE10A Q9Y233 2/20 0.36
PDE6D O43924 1/20 0.36
PDE6A P16499 1/20 0.36
PDE6G P18545 1/20 0.36
PDE6B P35913 1/20 0.36
PDE6C P51160 1/20 0.36
PDE6H Q13956 1/20 0.36
CYP1A2 P05177 2/20 0.35
PTGS2 P35354 1/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1B1 Q16678 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14183056 0.80 MEN1 (0.40) ACHEPOLBMEN1KMT2ALMNA
SCHEMBL684136 0.80 ACHE (0.52) ACHELMNAMAPTCYP3A4CA9
SCHEMBL15180051 0.77 POLB (0.39) ACHEPOLBMEN1KMT2ALMNA
SCHEMBL16838792 0.76 ALDH1A1 (0.42) POLBMEN1KMT2AMAPTCYP3A4
SCHEMBL18072590 0.76 MEN1 (0.50) POLBMEN1KMT2ALMNAMAPT
SCHEMBL14183048 0.76 MEN1 (0.47) POLBMEN1KMT2ALMNAMAPT
SCHEMBL4189560 0.75 MEN1 (0.36) POLBMEN1KMT2ALMNAMAPT
SCHEMBL27982688 0.72 POLB (0.36) POLBMEN1KMT2ALMNAMAPT
SCHEMBL19286922 0.72 ACHE (0.60) ACHEPOLBMEN1KMT2ALMNA
SCHEMBL21276080 0.71 MEN1 (0.39) ACHEPOLBMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012052420-A1 METHOD FOR PREPARING SUBSTITUTED N-(3-AMINO-QUINOXALIN-2-YL)-SULFONAMIDES AND THEIR INTERMEDIATES N-(3-CHLORO-QUINOXALIN-2-YL)SULFONAMIDES MERCK SERONO S.A. GENEVA (CH) 2012-04-26 WO disclosed