SCHEMBL10051978

SCHEMBL10051978

CC(C)(C)CNC(=O)c1cc(OCc2ccccc2)cc(-c2ccccc2)n1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.51
P2RY12 Q9H244 7/20 0.51
EGLN2 Q96KS0 1/20 0.45
EGLN1 Q9GZT9 1/20 0.45
ADORA2A P29274 2/20 0.42
ADORA1 P30542 2/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMPD1 P17405 1/20 0.41
SPHK2 Q9NRA0 1/20 0.41
SPHK1 Q9NYA1 1/20 0.41
XDH P47989 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10051977 0.82 CNR2 (0.46) P2RY12EGLN2ADORA2AADORA1MEN1
SCHEMBL4265711 0.81 MCL1 (0.74) MCL1P2RY12MEN1KMT2AXDH
SCHEMBL10052383 0.80 P2RY12 (0.50) P2RY12ADORA2AADORA1MEN1KMT2A
SCHEMBL4267162 0.77 MCL1 (0.58) MCL1P2RY12MEN1KMT2AXDH
SCHEMBL10052381 0.76 CNR2 (0.56) P2RY12
SCHEMBL10272688 0.74 HDAC3 (0.60) MEN1KMT2ASPHK2SPHK1
SCHEMBL4263343 0.72 MCL1 (0.52) MCL1P2RY12ADORA2AADORA1MEN1
SCHEMBL3534571 0.70 LMNA (0.55) MCL1MEN1KMT2A
SCHEMBL5035686 0.70 MAOB (0.59) MCL1MEN1KMT2A
SCHEMBL14278777 0.69 MEN1 (0.65) MCL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012019299-A1 HEPATITIS C INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-02-16 WO disclosed