SCHEMBL10053289

SCHEMBL10053289

COCOCc1ccc2c(c1)COB2c1cccc(C)c1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.31
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10053208 0.88 CYP3A4 (0.31) IDO1PDE4APDE4BPDE4CPDE4D
SCHEMBL10053282 0.81 PDE4A (0.34) PDE4APDE4BPDE4CPDE4D
SCHEMBL500011 0.74 CA1 (0.49) PDE4APDE4BPDE4CPDE4D
SCHEMBL10053280 0.73 CA1 (0.43) PDE4APDE4BPDE4CPDE4D
SCHEMBL16920264 0.71 IDO1 (0.58) IDO1MAOB
SCHEMBL10053224 0.69 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DMAOB
SCHEMBL21968362 0.68 IDO1 (0.55) IDO1MAOB
SCHEMBL21099587 0.68 IDO1 (0.55) IDO1MAOB
SCHEMBL10053299 0.66 ACHE (0.41) PDE4APDE4BPDE4CPDE4D
SCHEMBL10053203 0.66 PDE4B (0.34) PDE4APDE4BPDE4CPDE4DMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106031-B2 Hydrolytically-resistant boron-containing therapeutics and methods of use ANACOR PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed