SCHEMBL10053282

SCHEMBL10053282

Cc1cccc(B2OCc3cc(CO)ccc32)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
MAP2K4 P45985 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
PDE3A Q14432 1/20 0.31
PDCD1 Q15116 1/20 0.30
CD274 Q9NZQ7 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA7 P36544 1/20 0.30
CYP4F2 P78329 1/20 0.30
CYP4A11 Q02928 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10053283 0.85 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DCA1
SCHEMBL10053203 0.84 PDE4B (0.34) PDE4APDE4BPDE4CPDE4DCA1
SCHEMBL10053289 0.81 IDO1 (0.31) PDE4APDE4BPDE4CPDE4D
SCHEMBL500011 0.80 CA1 (0.49) PDE4APDE4BPDE4CPDE4DCA1
SCHEMBL597009 0.79 CA1 (0.49) PDE4APDE4BPDE4CPDE4DCA1
SCHEMBL10053280 0.79 CA1 (0.43) PDE4APDE4BPDE4CPDE4DCA1
SCHEMBL13996402 0.78 CA1 (0.44) CA1CA2CHRNB4CHRNA3CHRNA7
SCHEMBL10053224 0.74 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DCA1
SCHEMBL10053290 0.72 CA1 (0.31) PDE4APDE4BPDE4CPDE4DCA1
SCHEMBL10053299 0.71 ACHE (0.41) PDE4APDE4BPDE4CPDE4DCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106031-B2 Hydrolytically-resistant boron-containing therapeutics and methods of use ANACOR PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed