SCHEMBL10057504

SCHEMBL10057504

CC(C)(C)OC(=O)NC(Cc1ccccc1)C(=O)N[C@@H](CC(=O)N1CCCC1N)Cc1cc(F)c(F)cc1F

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.51
KLK5 Q9Y337 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CTSS P25774 4/20 0.46
CTSK P43235 3/20 0.46
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
F2 P00734 1/20 0.44
PRSS1 P07477 1/20 0.44
SCN9A Q15858 2/20 0.43
CMA1 P23946 4/20 0.43
CYP2D6 P10635 1/20 0.43
DPP4 P27487 1/20 0.43
DPP8 Q6V1X1 1/20 0.43
DPP9 Q86TI2 1/20 0.43
DPP7 Q9UHL4 1/20 0.43
REN P00797 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10057885 0.92 ACE (0.55) ACEKLK5L3MBTL1F2PRSS1
SCHEMBL572136 0.92 ACE (0.55) ACEKLK5L3MBTL1F2PRSS1
SCHEMBL572693 0.91 ACE (0.49) ACEKLK5L3MBTL1CTSSCTSK
SCHEMBL14982904 0.91 ACE (0.49) ACEKLK5L3MBTL1CTSSCTSK
SCHEMBL10057468 0.83 CTSS (0.54) ACEKLK5L3MBTL1CTSSCTSK
SCHEMBL571640 0.83 CTSS (0.54) ACEKLK5L3MBTL1CTSSCTSK
SCHEMBL571948 0.82 REN (0.53) ACEKLK5CTSSCTSKCTSL
SCHEMBL10057469 0.82 REN (0.53) ACEKLK5CTSSCTSKCTSL
SCHEMBL571617 0.80 CMA1 (0.57) ACEF2PRSS1CMA1
SCHEMBL10057884 0.80 CMA1 (0.57) ACEF2PRSS1CMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012017391-A2 NOVEL COMPOUNDS AS DPP-IV INHIBITORS AND PROCESS FOR PREPARATION THEREOF CADILA PHARMACEUTICALS LIMITED (IN) 2012-02-09 WO disclosed