SCHEMBL10059461

SCHEMBL10059461

Nc1cc(Br)ncc1NC1CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.43
HDAC1 Q13547 1/20 0.39
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
CDC42BPB Q9Y5S2 1/20 0.38
MAPK1 P28482 1/20 0.38
IGF1R P08069 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
PIM1 P11309 3/20 0.36
CYP1A2 P05177 3/20 0.34
BRD4 O60885 3/20 0.34
ATAD2 Q6PL18 3/20 0.34
CYP3A4 P08684 2/20 0.34
ALDH1A1 P00352 2/20 0.34
ALOX15 P16050 2/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 1/20 0.34
CYP2D6 P10635 1/20 0.34
KMT2A Q03164 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27171097 0.81 MAPK1 (0.44) HDAC1MAPK1HRH4
SCHEMBL617303 0.77 HRH3 (0.42) HRH3HDAC1ROCK2ROCK1CDC42BPB
SCHEMBL8244028 0.74 HRH3 (0.36) HRH3HDAC1ROCK2MAPK1IGF1R
SCHEMBL13808614 0.73 HRH3 (0.41) HRH3HDAC1ROCK2ROCK1CDC42BPB
SCHEMBL13742816 0.73 AOC1 (0.48) HRH3HDAC1ROCK2ROCK1CDC42BPB
SCHEMBL15740694 0.70 MEN1 (0.40) MAPK1MEN1CYP2D6KMT2ACYP2C19
SCHEMBL22725031 0.70 IKBKB (0.42) HRH3BRD4ATAD2CYP3A4ALDH1A1
SCHEMBL14046305 0.70 ROCK2 (0.50) HRH3ROCK2ROCK1CDC42BPBCYP1A2
Hydrochloric Acid SCHEMBL23360049 0.69 MAPK1 (0.47) HRH3ROCK2ROCK1CDC42BPBMAPK1
Hydrochloric Acid SCHEMBL29862503 0.69 MAPK1 (0.47) HRH3ROCK2ROCK1CDC42BPBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012086735-A1 CONDENSED HETEROCYCLIC COMPOUND 大正製薬株式会社 (JP) 2012-06-28 WO disclosed