SCHEMBL1006286

SCHEMBL1006286

c1ccc2c(CNC3CCNCC3)cccc2c1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.54
SLC6A2 P23975 1/20 0.54
SLC6A3 Q01959 1/20 0.54
CYP2D6 P10635 1/20 0.47
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.44
KMT2A Q03164 1/20 0.44
ACHE P22303 2/20 0.44
SOS1 Q07889 1/20 0.44
MC5R P33032 1/20 0.43
MC1R Q01726 1/20 0.43
CA2 P00918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2730868 0.89 ACHE (0.49) CYP2D6LMNAHTTKMT2AACHE
SCHEMBL15492796 0.85 HTT (0.55) LMNAHTTKMT2AACHECA2
SCHEMBL5767768 0.84 SLC6A2 (0.58) SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL10433983 0.84 KMT2A (0.57) LMNAHTTKMT2AACHE
SCHEMBL14194596 0.83 PRKCZ (0.51) SLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL10433976 0.83 KMT2A (0.56) LMNAHTTKMT2A
SCHEMBL8821304 0.78 TACR1 (0.50) SLC6A4SLC6A2SLC6A3
SCHEMBL14044360 0.78 SLC6A2 (0.52) SLC6A4SLC6A2SLC6A3LMNAHTT
SCHEMBL70402 0.78 SLC6A2 (0.52) SLC6A4SLC6A2SLC6A3LMNAHTT
SCHEMBL2779198 0.78 SLC6A2 (0.52) SLC6A4SLC6A2SLC6A3CYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268631-A1 AMINOPIPERIDINYL DERIVATIVES AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2011-01-05 EP disclosed
WO-2009118254-A1 AMINOPIPERIDINYL DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-10-01 WO disclosed