SCHEMBL10063155

SCHEMBL10063155

COc1ccc2c(c1)N(C1CCNCC1)C(=O)C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.45
CHRM4 P08173 3/20 0.45
CHRM5 P08912 3/20 0.45
CHRM1 P11229 3/20 0.45
CHRM3 P20309 3/20 0.45
HTR2C P28335 7/20 0.44
HTR2B P41595 5/20 0.44
HTR2A P28223 2/20 0.42
KYAT1 Q16773 1/20 0.40
KYAT3 Q6YP21 1/20 0.40
AADAT Q8N5Z0 1/20 0.40
HSD11B1 P28845 1/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
KMT2A Q03164 3/20 0.40
CASP1 P29466 1/20 0.40
GAA P10253 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15202987 0.92 HTR2C (0.51) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL982437 0.90 CHRM2 (0.49) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5872278 0.88 HTR2C (0.49) CHRM4CHRM1HTR2CHTR2BHTR2A
SCHEMBL10063157 0.82 CHRM2 (0.56) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL10063162 0.80 OPRM1 (0.40) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL10063525 0.78 BACE1 (0.55) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL3011324 0.77 HTR2A (0.42) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL26774954 0.77 PRKDC (0.62)
Hydrochloric Acid SCHEMBL3022954 0.76 HTR2A (0.41) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL828730 0.76 OPRM1 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020813-A1 FUSED-RING PYRROLIDINE DERIVATIVE 大日本住友製薬株式会社 (JP) 2012-02-16 WO disclosed