SCHEMBL10063533

SCHEMBL10063533

CCOC(=O)N1CCC(CN2CCC(N3C(=O)Cc4ccccc43)CC2)CC1

nearest known ligand 0.89

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.89
CHRM4 P08173 4/20 0.67
CHRM1 P11229 1/20 0.67
OPRM1 P35372 10/20 0.66
OPRL1 P41146 10/20 0.66
OPRK1 P41145 9/20 0.66
L3MBTL1 Q9Y468 1/20 0.55
HSD11B1 P28845 1/20 0.53
PLD1 Q13393 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15202958 0.94 KCNH2 (1.00) KCNH2CHRM4CHRM1OPRM1OPRL1
SCHEMBL15202998 0.92 KCNH2 (0.89) KCNH2CHRM4CHRM1OPRM1OPRL1
SCHEMBL10063163 0.86 KCNH2 (0.68) KCNH2CHRM4CHRM1OPRM1OPRL1
SCHEMBL10063524 0.85 KCNH2 (0.67) KCNH2CHRM4CHRM1OPRM1OPRL1
SCHEMBL13243464 0.83 KCNH2 (0.69) KCNH2CHRM4CHRM1OPRM1OPRL1
SCHEMBL2988260 0.83 KCNH2 (0.69) KCNH2CHRM4CHRM1OPRM1OPRL1
SCHEMBL13243461 0.83 KCNH2 (0.69) KCNH2CHRM4CHRM1OPRM1OPRL1
SCHEMBL7290423 0.82 KCNH2 (0.63) KCNH2L3MBTL1
SCHEMBL12791450 0.80 HSD11B1 (0.63) KCNH2CHRM4OPRM1OPRL1OPRK1
SCHEMBL1859950 0.80 OPRM1 (1.00) KCNH2OPRM1OPRL1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020813-A1 FUSED-RING PYRROLIDINE DERIVATIVE 大日本住友製薬株式会社 (JP) 2012-02-16 WO disclosed