SCHEMBL10065052

SCHEMBL10065052

CCCCOc1ccc2c(c1)c(I)c(C(=O)OCC)n2S(=O)(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 4/20 0.44
PSEN2 P49810 4/20 0.44
APH1B Q8WW43 4/20 0.44
NCSTN Q92542 4/20 0.44
APH1A Q96BI3 4/20 0.44
PSENEN Q9NZ42 4/20 0.44
ALDH1A1 P00352 1/20 0.44
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NOD2 Q9HC29 2/20 0.42
NOD1 Q9Y239 2/20 0.42
KAT6A Q92794 1/20 0.42
PTGDR Q13258 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2005697 0.85 NOD2 (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL10065051 0.82 PSEN1 (0.40) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL10064904 0.78 PSEN1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2343252 0.77 HTR6 (0.50) TP53KMT2ANOD2NOD1PTGDR
SCHEMBL2731882 0.76 HTR6 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2344679 0.76 NOD2 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL10064902 0.75 PSEN1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2540534 0.73 NOD2 (0.53) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2345728 0.73 NOD2 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2346812 0.73 NOD2 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059568-A1 NOVEL WATER-SOLUBLE INDOLOBENZAZEPINE MOLECULES DEMONSTRATING ANTIMITOTIC, ANTIVASCULAR, AND ANTITUMOR ACTIVITIES IN VIVO CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2012-05-10 WO disclosed