Stearylsulfamide

Stearylsulfamide

SCHEMBL1006541

CCCCCCCCCCCCCCCCCC(=O)NS(=O)(=O)c1ccc(N)cc1.[NaH]

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.57
TSHR P16473 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
EPHX2 P34913 1/20 0.54
DHFR P00374 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
MAPT P10636 1/20 0.51
CA12 O43570 2/20 0.49
CA9 Q16790 2/20 0.49
RAB9A P51151 2/20 0.48
KMT2A Q03164 2/20 0.48
FBP1 P09467 1/20 0.46
LMNA P02545 2/20 0.46
MEN1 O00255 1/20 0.46
ALB P02768 1/20 0.45
CYP2C9 P11712 1/20 0.45
AKT1 P31749 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Stearylsulfamide SCHEMBL15335 0.99 ALDH1A1 (0.58) ALDH1A1TSHRTDP1EPHX2DHFR
SCHEMBL107968 0.99 ALDH1A1 (0.58) ALDH1A1TSHRTDP1EPHX2DHFR
Stearylsulfamide SCHEMBL17981340 0.99 ALDH1A1 (0.58) ALDH1A1TSHRTDP1EPHX2DHFR
Stearylsulfamide SCHEMBL5731325 0.99 ALDH1A1 (0.58) ALDH1A1TSHRTDP1EPHX2DHFR
Stearylsulfamide SCHEMBL7162273 0.97 ALDH1A1 (0.55) ALDH1A1TSHRTDP1EPHX2DHFR
Stearylsulfamide SCHEMBL4663113 0.97 ALDH1A1 (0.57) ALDH1A1TSHRTDP1EPHX2DHFR
Stearylsulfamide SCHEMBL9070453 0.97 ALDH1A1 (0.57) ALDH1A1TSHRTDP1EPHX2DHFR
Stearylsulfamide SCHEMBL2714792 0.97 ALDH1A1 (0.57) ALDH1A1TSHRTDP1EPHX2DHFR
Stearylsulfamide SCHEMBL322075 0.97 ALDH1A1 (0.57) ALDH1A1TSHRTDP1EPHX2DHFR
Stearylsulfamide SCHEMBL2367792 0.97 ALDH1A1 (0.57) ALDH1A1TSHRTDP1EPHX2DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 132 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223821-A1 PROCESS FOR CHEMICALS AND ENERGY RECOVERY. CROON INVENTOR (SE) 1987-06-03 EP claimed
WO-1986007396-A1 PROCESS FOR CHEMICALS AND ENERGY RECOVERY CROON INVENTOR AKTIEBOLAG (SE) 1986-12-18 WO claimed
WO-2023220131-A2 PI3Kα INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2023-11-16 WO disclosed
EP-3915977-A1 1,2,3,4-TETRAHYDROQUINOXALINE DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Abbisko Therapeutics Co., Ltd. (CN) 2021-12-01 EP disclosed
EP-3653613-A1 1,3-DI-SUBSTITUTED KETENE COMPOUND AND APPLICATION THEREOF Guangzhou Bebetter Medicine Technology Co., Ltd. (CN) 2020-05-20 EP disclosed
EP-3519057-A1 A METHOD OF TREATING A MATERIAL COMPRISING AN AMINE SALT OF A CARBOXYLIC ACID HAVING 4 TO 10 CARBON ATOMS Innospec Limited (GB) 2019-08-07 EP disclosed
EP-3481430-A1 NUCLEIC ACID CONJUGATES AND USES THEREOF TRANSLATE BIO MA, INC. (US) 2019-05-15 EP disclosed
WO-2018060719-A1 A METHOD OF TREATING A MATERIAL COMPRISING AN AMINE SALT OF A CARBOXYLIC ACID HAVING 4 TO 10 CARBON ATOMS INNOSPEC LIMITED (GB) 2018-04-05 WO disclosed
WO-2018013525-A1 NUCLEIC ACID CONJUGATES AND USES THEREOF TRANSLATE BIO MA, INC. (US) 2018-01-18 WO disclosed
WO-2017182819-A1 METHODS, COMPOSITIONS AND USES RELATING THERETO INNOSPEC LIMITED (GB) 2017-10-26 WO disclosed
EP-2822928-A1 SUBSTITUTED HETEROCYCLIC ACETAMIDES AS KAPPA OPIOID RECEPTOR (KOR) AGONISTS Dr. Reddy's Laboratories Ltd. (IN) 2015-01-14 EP disclosed
WO-1989003024-A1 APPARATUS AND METHOD FOR IMAGING AND COUNTING MOVING PARTICLES QUADTEK, INC. (US) 1989-04-06 WO disclosed
EP-0229053-A1 METHOD FOR SYNTHESIZING DEOXYOLIGONUCLEOTIDES UNIVERSITY PATENTS, INC. (US) 1987-07-22 EP disclosed
WO-1986007362-A1 METHOD FOR SYNTHESIZING DEOXYOLIGONUCLEOTIDES UNIVERSITY PATENTS, INC. (US) 1986-12-18 WO disclosed
EP-0128937-A1 DRUG ABUSE TEST INDICATOR DEVICE AND METHOD OF MAKING SAME MEDICAL DIAGNOSTICS INC. (US) 1984-12-27 EP disclosed
WO-1984002397-A1 DRUG ABUSE TEST INDICATOR DEVICE AND METHOD OF MAKING SAME MEDICAL DIAGNOSTICS INC (US) 1984-06-21 WO disclosed
EP-0070170-A1 Tylosin derivatives, their preparation and pharmaceutical compositions containing them ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1983-01-19 EP disclosed
EP-0060258-A4 METHOD FOR PRODUCING 3,6-BIS(CARBOETHOXYAMINO)-2,5-DIAZIRIDINYL-1,4-BENZOQUINONE. AEROJET GENERAL CO (US) 1982-12-02 EP disclosed
EP-0060258-A1 METHOD FOR PRODUCING 3,6-BIS(CARBOETHOXYAMINO)-2,5-DIAZIRIDINYL-1,4-BENZOQUINONE. AEROJET GENERAL CO (US) 1982-09-22 EP disclosed
WO-1982000823-A1 METHOD FOR PRODUCING 3,6-BIS(CARBOETHOXYAMINO)-2,5-DIAZIRIDINYL-1,4-BENZOQUINONE AEROJET GENERAL CO (US) 1982-03-18 WO disclosed