SCHEMBL10065869

SCHEMBL10065869

Cc1ccc(N=O)cc1Nc1ncc(-c2ccncc2)o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 6/20 0.46
ALOX5 P09917 1/20 0.44
KDR P35968 9/20 0.42
FLT1 P17948 8/20 0.42
FLT4 P35916 8/20 0.42
TRPV1 Q8NER1 1/20 0.41
IMPDH2 P12268 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
STAT1 P42224 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
P2RY1 P47900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2346410 0.86 KIT (0.44) KITALOX5KDRFLT1FLT4
SCHEMBL10066362 0.85 FLT1 (0.51) KITALOX5KDRFLT1FLT4
SCHEMBL2339077 0.82 KIT (0.48) KITALOX5KDRFLT1FLT4
SCHEMBL2828692 0.80 FLT1 (0.49) KITALOX5KDRFLT1FLT4
SCHEMBL2343342 0.80 ALDH1A1 (0.47) KITALOX5KDRFLT1FLT4
SCHEMBL544406 0.80 IMPDH2 (0.62) KITKDRFLT1FLT4IMPDH2
SCHEMBL543637 0.79 FLT1 (0.44) KITALOX5KDRFLT1FLT4
SCHEMBL16365782 0.79 KIT (0.51) KITALOX5KDRFLT1FLT4
SCHEMBL543854 0.77 IMPDH2 (0.56) KITKDRFLT1FLT4IMPDH2
SCHEMBL13380736 0.76 KIT (0.43) KITALOX5KDRFLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120108616-A1 SUBSTITUTED OXAZOLE DERIVATIVES AND THEIR USE AS TYROSINE KINASE INHIBITORS AB SCIENCE 2012-05-03 US disclosed
US-20080242704-A1 Substituted Oxazole Derivatives and their Use as Tyrosine Kinase Inhibitors AB SCIENCE 2008-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242704-A1 Substituted Oxazole Derivatives and their Use as Tyrosine Kinase Inhibitors KIT, TYRO3, LCK KIT 1/4885ALOX5 3096/4885KDR 240/4885
US-20120108616-A1 SUBSTITUTED OXAZOLE DERIVATIVES AND THEIR USE AS TYROSINE KINASE INHIBITORS KIT, FLT3, LTK KIT 1/4885ALOX5 2289/4885KDR 36/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.