SCHEMBL10066580

SCHEMBL10066580

CCc1cccc(-c2ncn[nH]2)c1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.58
ENPP2 Q13822 1/20 0.58
MRGPRX4 Q96LA9 1/20 0.49
NOTUM Q6P988 1/20 0.47
NISCH Q9Y2I1 1/20 0.45
EGFR P00533 1/20 0.44
FGFR1 P11362 1/20 0.41
BCL2 P10415 1/20 0.41
LRRK2 Q5S007 1/20 0.39
PTGS2 P35354 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10066946 0.79 METAP2 (0.44) IDO1ENPP2NOTUMNISCH
SCHEMBL8136764 0.78 ENPP2 (0.55) IDO1ENPP2NOTUMEGFRFGFR1
SCHEMBL16168686 0.77 IDO1 (0.64) IDO1ENPP2NOTUMNISCHEGFR
SCHEMBL22501795 0.75 ENPP2 (0.52) IDO1ENPP2MRGPRX4EGFR
SCHEMBL5378711 0.74 MAPK8 (0.54) IDO1ENPP2MRGPRX4EGFRFGFR1
SCHEMBL1334565 0.74 IDO1 (1.00) IDO1ENPP2MRGPRX4NOTUM
SCHEMBL1985682 0.74 IDO1 (0.64) IDO1ENPP2MRGPRX4EGFR
SCHEMBL3080603 0.74 ENPP2 (1.00) IDO1ENPP2
SCHEMBL2659146 0.74 IDO1 (0.64) IDO1ENPP2
SCHEMBL179125 0.73 NISCH (0.55) IDO1MRGPRX4NOTUMNISCHFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006203-A1 N-CYCLYL-3 - (CYCLYLCARBONYLAMINOMETHYL) BENZAMIDE DERIVATIVES AS RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-12 WO disclosed