SCHEMBL10067701

SCHEMBL10067701

CC(C)[C@@H](Nc1ccnc(C2CNc3ncc(Cl)cc32)n1)C(=O)NCCC(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTRA1 Q92743 8/20 0.33
IDO1 P14902 1/20 0.31
MAPK1 P28482 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.30
IDH1 O75874 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13060106 0.87 IDH1 (0.31) IRAK4IDH1
SCHEMBL10067630 0.87 TRPV3 (0.31) IDH1
SCHEMBL10067629 0.87 TRPV3 (0.31) IDH1
SCHEMBL10067942 0.86 IDH1 (0.31) IDH1
SCHEMBL13060037 0.85
SCHEMBL2633646 0.85
SCHEMBL2633775 0.84 MAPK1 (0.34) MAPK1
SCHEMBL13059455 0.83 BTK (0.35) IRAK4IDH1
SCHEMBL13060039 0.82 ULK1 (0.32) HTRA1IDO1
SCHEMBL10068280 0.81 JAK1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163917-B2 Azaindoles useful as inhibitors of Janus kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-04-24 US disclosed