SCHEMBL10067975

SCHEMBL10067975

O=C(NC[C@@H]1CCCO1)c1nc(-c2nnnn2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
GSK3B P49841 2/20 0.44
KCNH2 Q12809 1/20 0.44
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
HPGD P15428 8/20 0.42
GAA P10253 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HTT P42858 1/20 0.40
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067976 0.85 GSK3B (0.44) ALDH1A1GSK3BKCNH2RAB9ANPC1
SCHEMBL14600774 0.85 GSK3B (0.45) ALDH1A1GSK3BKCNH2RAB9ANPC1
SCHEMBL14278771 0.84 MAPK1 (0.49) ALDH1A1GSK3BKCNH2RAB9ANPC1
SCHEMBL10067977 0.83 GSK3B (0.47) GSK3BKCNH2RAB9ANPC1HPGD
SCHEMBL14600763 0.81 GSK3B (0.44) ALDH1A1GSK3BKCNH2RAB9ANPC1
SCHEMBL10067973 0.80 RAB9A (0.51) ALDH1A1GSK3BKCNH2RAB9ANPC1
SCHEMBL14600765 0.78 ADORA2A (0.41) RAB9ANPC1KMT2AMEN1
SCHEMBL14286176 0.77 HPGD (0.52) ALDH1A1HPGDGAACYP1A2CYP2C9
SCHEMBL14600777 0.77 GSK3B (0.53) ALDH1A1GSK3BKCNH2RAB9ANPC1
SCHEMBL14600753 0.76 GSK3B (0.53) ALDH1A1GSK3BKCNH2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697352-B1 4-AZOLE SUBSTITUTED IMIDAZOLE COMPOSITIONS USEFUL AS INHIBITORS OR C-MET RECEPTOR TYROSINE KINASE VERTEX PHARMA (US) 2012-06-27 EP disclosed
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed