SCHEMBL10068629

SCHEMBL10068629

C=C1O[C@@H](COP(=O)(O)O)CN1c1ccc(-c2ccc(N3CCNC3=O)nc2)c(F)c1F

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.41
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
CNR2 P34972 1/20 0.32
CETP P11597 3/20 0.32
CALML3 P27482 1/20 0.31
MAOA P21397 4/20 0.31
ROCK2 O75116 2/20 0.31
MAOB P27338 2/20 0.31
MGLL Q99685 1/20 0.31
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
ALK Q9UM73 1/20 0.30
GRM5 P41594 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL412646 0.93 TDO2 (0.42) TDO2CETPCALML3MAOAMAOB
SCHEMBL469913 0.87 CALML3 (0.44) TDO2CALML3MAOAMAOBCYP2C9
SCHEMBL10068630 0.85 TDO2 (0.42) TDO2CETPCALML3MAOAMAOB
SCHEMBL412829 0.81 CALML3 (0.53) CALML3MAOAMAOBCYP2C9CYP2C19
SCHEMBL412791 0.80 GRM5 (0.36) CNR2CALML3MAOAMAOBCYP2C9
SCHEMBL412753 0.80 CALML3 (0.48) TDO2CALML3MAOAMAOBCYP2C9
SCHEMBL412640 0.79 TDO2 (0.43) TDO2CALML3MAOAMAOBCYP2C9
SCHEMBL412794 0.79 TDO2 (0.46) TDO2CALML3MAOAMAOBCYP2C9
SCHEMBL411159 0.79 TDO2 (0.39) TDO2CALML3MAOAMAOBCYP2C9
SCHEMBL411080 0.78 TDO2 (0.40) TDO2CALML3MAOAMAOBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033952-A1 3 - PHENYL- 2 -OXO- 1, 3 -OXAZOLIDINES FOR TREATMENT OF BACTERIAL INFECTIONS MICURX PHARMACEUTICALS, INC. (KY) 2012-03-15 WO disclosed