SCHEMBL469913

SCHEMBL469913

C=C1O[C@@H](COP(=O)(O)O)CN1c1ccc(-c2ccc(N3CCNC3=O)nc2)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CALML3 P27482 4/20 0.44
TDO2 P48775 1/20 0.43
MAOA P21397 14/20 0.42
MAOB P27338 2/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL412829 0.93 CALML3 (0.53) CALML3MAOAMAOBCYP2C9CYP2C19
SCHEMBL10068630 0.92 TDO2 (0.42) CALML3TDO2MAOAMAOBCYP2C9
SCHEMBL10068629 0.87 TDO2 (0.41) CALML3TDO2MAOAMAOBCYP2C9
SCHEMBL412640 0.84 TDO2 (0.43) CALML3TDO2MAOAMAOBCYP2C9
SCHEMBL10069650 0.83 MAOA (0.43) CALML3TDO2MAOAMAOBCYP2C19
SCHEMBL411159 0.82 TDO2 (0.39) CALML3TDO2MAOAMAOBCYP2C9
SCHEMBL412646 0.81 TDO2 (0.42) CALML3TDO2MAOAMAOBCYP2C9
SCHEMBL411105 0.81 CALML3 (0.51) CALML3MAOAMAOBCYP2C9CYP2C19
SCHEMBL411061 0.81 MAOA (0.51) CALML3MAOAMAOBCYP2C9CYP2C19
SCHEMBL411603 0.81 CALML3 (0.50) CALML3MAOAMAOBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033952-A1 3 - PHENYL- 2 -OXO- 1, 3 -OXAZOLIDINES FOR TREATMENT OF BACTERIAL INFECTIONS MICURX PHARMACEUTICALS, INC. (KY) 2012-03-15 WO disclosed