SCHEMBL1006876

SCHEMBL1006876

CCC(C)Oc1ccc2c(n1)c(N)nc1ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 13/20 0.48
TLR8 Q9NR97 10/20 0.48
ADORA2A P29274 6/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
HRH2 P25021 1/20 0.42
ADRA1D P25100 1/20 0.42
HTR2A P28223 1/20 0.42
ADRA1A P35348 1/20 0.42
NUDT1 P36639 1/20 0.42
HTR2B P41595 1/20 0.42
PDE4D Q08499 1/20 0.42
KCNH2 Q12809 1/20 0.42
ADORA3 P0DMS8 5/20 0.42
ADORA1 P30542 4/20 0.42
MCHR1 Q99705 1/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1007829 0.78 ADORA2A (0.53) TLR7TLR8ADORA2APOLBADRA1A
SCHEMBL1061503 0.77 TLR8 (0.55) TLR7TLR8ADORA2AADORA3ADORA1
SCHEMBL1006095 0.73 ADORA1 (0.49) TLR7TLR8ADORA2ANUDT1ADORA3
SCHEMBL17054092 0.73 GPBAR1 (0.53) TLR8LMNAMCHR1GABRPGABRD
SCHEMBL1010427 0.72 TLR7 (0.57) TLR7TLR8ADORA2ALMNAPOLB
SCHEMBL1009385 0.72 TLR7 (0.54) TLR7TLR8ADORA2ALMNAPOLB
SCHEMBL1703456 0.71 TLR7 (0.57) TLR7TLR8ADORA2ALMNAPOLB
SCHEMBL1675410 0.71 ADORA3 (0.43) TLR7TLR8ADORA2AADORA3ADORA1
SCHEMBL1008185 0.70 TLR7 (0.54) TLR7TLR8ADORA2AADRA1ANUDT1
SCHEMBL1008581 0.69 TLR7 (0.52) TLR7TLR8ADORA2ANUDT1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268618-A1 COMPOUNDS AND COMPOSITIONS AS TLR ACTIVITY MODULATORS IRM LLC (BM) 2011-01-05 EP disclosed