SCHEMBL10068784

SCHEMBL10068784

COCCOc1cc(C(=O)O)cc(C(OCCNC(=O)OC)c2cccc(Cl)c2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
HTT P42858 3/20 0.39
MAPT P10636 2/20 0.39
LMNA P02545 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GCK P35557 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TSHR P16473 2/20 0.38
MAPK1 P28482 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTR1A P08908 1/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
ADRB3 P13945 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10068952 0.95 HTT (0.38) MEN1KMT2AHTTMAPTLMNA
SCHEMBL10068802 0.93 KLKB1 (0.41) MEN1KMT2AHTTMAPTLMNA
SCHEMBL10068767 0.92 FAAH (0.43) KMT2AMAPTSMN1; SMN2ADRB3ALDH1A1
SCHEMBL10068721 0.92 HTT (0.40) MEN1KMT2AHTTMAPTLMNA
SCHEMBL10069328 0.91 ADRB3 (0.42) MEN1KMT2AHTTMAPTLMNA
SCHEMBL10069339 0.90 KDM4E (0.47) MEN1KMT2AHTTMAPTLMNA
SCHEMBL10068561 0.90 TSHR (0.45) MEN1KMT2AHTTMAPTLMNA
SCHEMBL10068546 0.88 HTT (0.36) MEN1KMT2AHTTMAPTLMNA
SCHEMBL2027362 0.88 HTT (0.43) MEN1KMT2AHTTMAPTLMNA
SCHEMBL10068953 0.88 KLKB1 (0.40) MEN1KMT2AHTTMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012019428-A1 BENZOHYDROL DERIVATIVES, A PREPARATION PROCESS AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-02-16 WO disclosed