SCHEMBL10069253

SCHEMBL10069253

CC(=O)[C@@H](N)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 10/20 0.54
SLC22A2 O15244 1/20 0.52
SLC47A1 Q96FL8 1/20 0.52
MAPT P10636 1/20 0.50
ALDH1A1 P00352 2/20 0.48
NPC1 O15118 1/20 0.48
FAP Q12884 1/20 0.44
PITRM1 Q5JRX3 1/20 0.44
DPP8 Q6V1X1 1/20 0.44
DPP9 Q86TI2 1/20 0.44
DPP7 Q9UHL4 1/20 0.44
CYP3A4 P08684 1/20 0.43
THRB P10828 1/20 0.41
CYP2C9 P11712 1/20 0.41
EPHX1 P07099 1/20 0.40
EPHX2 P34913 1/20 0.39
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2623068 0.81 DPP4 (0.61) DPP4FAPPITRM1DPP8DPP9
SCHEMBL255570 0.80 DPP4 (0.49) DPP4SLC22A2SLC47A1MAPTALDH1A1
SCHEMBL23460047 0.80 DPP4 (0.49) DPP4SLC22A2SLC47A1MAPTALDH1A1
SCHEMBL18397921 0.80 ALDH1A1 (0.50) DPP4SLC22A2SLC47A1MAPTALDH1A1
SCHEMBL6739912 0.80 DPP4 (0.49) DPP4SLC22A2SLC47A1MAPTALDH1A1
Hydrochloric Acid SCHEMBL28561377 0.78 ALDH1A1 (0.50) DPP4SLC22A2SLC47A1MAPTALDH1A1
Hydrochloric Acid SCHEMBL28561376 0.78 ALDH1A1 (0.50) DPP4SLC22A2SLC47A1MAPTALDH1A1
SCHEMBL15535092 0.78 DPP4 (0.51) DPP4SLC22A2SLC47A1MAPTALDH1A1
SCHEMBL15149731 0.78 DPP4 (0.51) DPP4SLC22A2SLC47A1MAPTALDH1A1
SCHEMBL8073575 0.76 ALDH1A1 (0.50) DPP4SLC22A2SLC47A1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021876-A2 PEPTIDOMIMETIC MACROCYCLES AILERON THERAPEUTICS, INC. (US) 2012-02-16 WO disclosed