SCHEMBL10070429

SCHEMBL10070429

CCCCOc1c(C(=O)OC)nc2c(N(C)SC)cc(N3CCN(C)CC3)cn2c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SIRT6 Q8N6T7 1/20 0.32
LCK P06239 1/20 0.31
SRC P12931 1/20 0.31
GAA P10253 2/20 0.31
HRH4 Q9H3N8 1/20 0.31
HDAC3 O15379 2/20 0.31
HDAC8 Q9BY41 2/20 0.31
FGFR3 P22607 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
EGFR P00533 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
MTOR P42345 1/20 0.30
MMP1 P03956 1/20 0.30
MMP9 P14780 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10071002 0.92 TSHR (0.36) HPGDMAPTTSHRTAAR1HSD17B10
SCHEMBL15101327 0.89 MAPT (0.35) HPGDMAPTTSHRTAAR1HSD17B10
SCHEMBL10070043 0.82 TSHR (0.35) HPGDMAPTTSHRTAAR1HSD17B10
SCHEMBL10070052 0.81 TSHR (0.35) HPGDMAPTTSHRTAAR1HSD17B10
SCHEMBL10070064 0.81 HPGD (0.35) HPGDMAPTTSHRTAAR1HSD17B10
SCHEMBL10070425 0.81 SYK (0.40) HPGDMAPTTSHRTAAR1HSD17B10
SCHEMBL10070066 0.81 MAPT (0.37) HPGDMAPTHSD17B10KDM4EALDH1A1
SCHEMBL10070068 0.80 HSD17B10 (0.35) HPGDMAPTTSHRTAAR1HSD17B10
SCHEMBL10069878 0.80 HPGD (0.35) HPGDMAPTTSHRTAAR1HSD17B10
SCHEMBL15101373 0.80 MET (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006680-A1 7, 9-NITROGEN RADICAL-4-OXO-4H-PYRIDO[L,2-A]PYRIMIDINE-2-CARBOXYLIC ACID BENZYLAMIDE ANTI-VIRALS AVEXA LIMITED (AU) 2012-01-19 WO disclosed