SCHEMBL10071006

SCHEMBL10071006

CCCCCN(C=O)c1cc(N2CCN(C)CC2)cn2c(=O)c(O)c(C(=O)NCc3ccc(F)cc3)nc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
KCNH2 Q12809 1/20 0.39
POLB P06746 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
ACE2 Q9BYF1 1/20 0.37
CCR1 P32246 2/20 0.36
KCNE1 P15382 1/20 0.36
KCNQ1 P51787 1/20 0.36
TTK P33981 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KMT2A Q03164 1/20 0.35
CALCA P06881 1/20 0.35
DCTPP1 Q9H773 2/20 0.34
ENPP2 Q13822 1/20 0.34
ERCC1 P07992 1/20 0.34
FEN1 P39748 1/20 0.34
ERCC4 Q92889 1/20 0.34
SMO Q99835 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL359611 0.83 KCNH2 (0.46) CYP2C9CYP3A4CYP2C19KCNH2POLB
SCHEMBL826461 0.78 CYP2C9 (0.45) CYP2C9CYP3A4CYP2C19KCNH2CCR1
SCHEMBL826251 0.78 CYP2C9 (0.54) CYP2C9CYP3A4CYP2C19KCNH2ACE2
SCHEMBL10069921 0.78 CALCA (0.41) CYP2C9CYP3A4CYP2C19KCNH2POLB
SCHEMBL368651 0.77 LMNA (0.45) CYP2C9CYP3A4CYP2C19KCNH2ACE2
SCHEMBL368831 0.77 KCNH2 (0.42) CYP2C9CYP3A4CYP2C19KCNH2POLB
SCHEMBL371233 0.77 LMNA (0.47) CYP2C9CYP3A4CYP2C19KCNH2ACE2
SCHEMBL10070414 0.77 CNR2 (0.39) CYP2C9CYP3A4CYP2C19KCNH2POLB
SCHEMBL369169 0.77 ACE2 (0.41) CYP2C9CYP3A4CYP2C19KCNH2ACE2
SCHEMBL359557 0.76 CYP2C9 (0.43) CYP2C9CYP3A4CYP2C19KCNH2CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006680-A1 7, 9-NITROGEN RADICAL-4-OXO-4H-PYRIDO[L,2-A]PYRIMIDINE-2-CARBOXYLIC ACID BENZYLAMIDE ANTI-VIRALS AVEXA LIMITED (AU) 2012-01-19 WO disclosed