SCHEMBL282170

SCHEMBL282170

CCc1cc(NC(=O)Nc2ccc(Oc3ncnc4cc(F)c(C)cc34)cc2)ccc1Cl

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.62
CSF1R P07333 7/20 0.53
PDGFRA P16234 1/20 0.53
FLT1 P17948 1/20 0.49
FLT4 P35916 1/20 0.49
BRAF P15056 2/20 0.49
RAF1 P04049 1/20 0.49
MAPK14 Q16539 1/20 0.49
TNNI3K Q59H18 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL281945 0.86 KDR (0.57) KDRCSF1RPDGFRABRAFRAF1
SCHEMBL10073792 0.85 CSF1R (0.73) KDRCSF1RPDGFRAFLT1FLT4
SCHEMBL282171 0.80 RAF1 (0.44) KDRPDGFRABRAFRAF1
SCHEMBL281804 0.76 KDR (0.70) KDRPDGFRA
SCHEMBL282308 0.73 CSF1R (0.70) KDRCSF1RPDGFRABRAFRAF1
SCHEMBL17668250 0.72 BRAF (0.81) KDRPDGFRABRAFRAF1
SCHEMBL26894919 0.72 KDR (0.71) KDRPDGFRAFLT1FLT4BRAF
SCHEMBL5202980 0.72 KDR (0.85) KDRCSF1RPDGFRAFLT1FLT4
SCHEMBL7480612 0.70 KDR (1.00) KDRCSF1RPDGFRAFLT1FLT4
SCHEMBL10073787 0.70 CSF1R (1.00) KDRCSF1RFLT1FLT4BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2428506-A1 HETEROCYCLIC SUBSTITUTED ACARDITE DERIVATES AND USE THEREOF Jiangsu Provincial Institute Of Materia Medica Co. (CN) 2012-03-14 EP claimed
US-20120053192-A1 Heterocyclic Substituted Acardite Derivate and Application Thereof NANJING LUYESIKE PHARMACEUTICAL CO., LTD. (CN) 2012-03-01 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120053192-A1 Heterocyclic Substituted Acardite Derivate and Application Thereof H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, IDH1, CA7 KDR 3633/4885CSF1R 2180/4885PDGFRA 1115/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.