SCHEMBL10074338

SCHEMBL10074338

Cc1cccc(-c2cc(C#N)ccc2C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.44
ADORA1 P30542 2/20 0.44
CYP11B1 P15538 2/20 0.44
CYP11B2 P19099 2/20 0.44
AR P10275 2/20 0.43
LRRK2 Q5S007 2/20 0.42
KDM4E B2RXH2 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
MAPK14 Q16539 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP2A6 P11509 1/20 0.41
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ABL1 P00519 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16429408 0.86 EGLN2 (0.46) ADORA2AADORA1CYP11B1CYP11B2AR
SCHEMBL18406712 0.85 AR (0.51) ADORA2AADORA1CYP11B1CYP11B2AR
SCHEMBL15856481 0.84 PTGDR2 (0.49) CYP11B1CYP11B2ARKDM4ECYP1A2
SCHEMBL29788076 0.84 PTGDR2 (0.49) CYP11B1CYP11B2ARKDM4ECYP1A2
SCHEMBL18406706 0.81 AR (0.48) ADORA2AADORA1CYP11B1CYP11B2AR
SCHEMBL5099548 0.81 PLAU (0.46) ADORA2AADORA1ARLRRK2KDM4E
SCHEMBL7386770 0.80 CLK4 (0.53) ARKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL18934331 0.80 ALDH1A1 (0.54) CYP11B1CYP11B2ARALDH1A1CYP2A6
SCHEMBL278217 0.79 S1PR4 (0.53) ADORA1LRRK2MAPTHPGDTSHR
SCHEMBL6110387 0.78 AR (0.54) CYP11B1CYP11B2ARMAPK14ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012022045-A1 PYRROLOPYRIMIDINE COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2012-02-23 WO disclosed