SCHEMBL10076664

SCHEMBL10076664

CN1C(=O)CCNc2ccc(C(F)(F)F)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.44
PARP1 P09874 1/20 0.44
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
BRPF1 P55201 1/20 0.39
AR P10275 1/20 0.39
TRPV1 Q8NER1 2/20 0.38
SRD5A1 P18405 1/20 0.37
KIF11 P52732 3/20 0.37
HSP90AA1 P07900 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2628423 0.82 PARP10 (0.42) PARP10PARP1KMT2AMEN1MAPT
SCHEMBL31470006 0.76 MAPT (0.49) PARP10PARP1KMT2AMEN1MAPT
SCHEMBL5230478 0.73 BRPF1 (0.69) PARP10PARP1KMT2AMEN1MAPT
SCHEMBL31020734 0.72 KMT2A (0.51) KMT2AMEN1MAPTALDH1A1GAA
SCHEMBL14288738 0.71 MAPT (0.44) KMT2AMEN1MAPTALDH1A1MAPK1
SCHEMBL12894753 0.71 PARP10 (0.58) PARP10PARP1KMT2AMEN1MAPT
SCHEMBL11425719 0.70 PARP10 (0.41) PARP10PARP1KMT2AMEN1MAPT
SCHEMBL2632664 0.70 KIF11 (0.54) PARP10PARP1KIF11
SCHEMBL4991137 0.70 PARP10 (0.56) PARP10PARP1GAAARKIF11
SCHEMBL11419524 0.69 MEN1 (0.51) KMT2AMEN1MAPTALDH1A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418213-A1 NEUROMEDIN U DERIVATIVE Takeda Pharmaceutical Company Limited (JP) 2012-02-15 EP disclosed