SCHEMBL10078403

SCHEMBL10078403

NC(=O)C(=O)c1c[nH]c2cccc(F)c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.49
GPR84 Q9NQS5 2/20 0.49
FFAR1 O14842 1/20 0.49
ALDH1A1 P00352 1/20 0.45
ATM Q13315 1/20 0.45
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
IGF1R P08069 1/20 0.42
SRC P12931 1/20 0.42
ALB P02768 1/20 0.41
IL2 P60568 1/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 1/20 0.41
NR4A2 P43354 1/20 0.41
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10321304 0.88 ALDH1A1 (0.54) HTR2AGPR84FFAR1ALDH1A1ATM
SCHEMBL1558360 0.87 HTR2A (0.49) HTR2AGPR84FFAR1ALDH1A1ATM
SCHEMBL1732171 0.85 HTR2A (0.47) HTR2AGPR84FFAR1ALDH1A1ATM
SCHEMBL10083723 0.85 HTR2A (0.47) HTR2AGPR84FFAR1ALDH1A1ATM
SCHEMBL2034897 0.83 GPR84 (0.51) HTR2AGPR84FFAR1ALDH1A1GAA
SCHEMBL14363141 0.81 HTR2A (0.48) HTR2AGPR84FFAR1ALDH1A1ATM
SCHEMBL25678359 0.81 HTR2A (0.47) HTR2AGPR84FFAR1ALDH1A1ATM
SCHEMBL23160620 0.81 GPR84 (0.50) HTR2AGPR84FFAR1ALDH1A1ATM
SCHEMBL16234666 0.81 PBRM1 (0.54) HTR2AGPR84FFAR1IGF1RSRC
SCHEMBL3721316 0.80 GPR84 (0.49) HTR2AGPR84ALDH1A1ATMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013170-B1 4-SQUARYLPIPERAZINE DERIVATIVES AS ANTIVIRAL AGENTS BRISTOL MYERS SQUIBB CO (US) 2012-06-27 EP disclosed