SCHEMBL10079015

SCHEMBL10079015

CC(=O)[C@@H](N)Cc1c[nH]c2cc(Cl)ccc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.57
GPR84 Q9NQS5 1/20 0.55
SOS1 Q07889 7/20 0.54
PTPRA P18433 1/20 0.51
KDM4E B2RXH2 2/20 0.50
LMNA P02545 2/20 0.50
MAPT P10636 2/20 0.50
TSHR P16473 2/20 0.50
BLM P54132 2/20 0.50
PMP22 Q01453 2/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
MPO P05164 1/20 0.50
HIF1A Q16665 1/20 0.50
CYP2C19 P33261 1/20 0.49
ADRB3 P13945 1/20 0.48
SLC6A4 P31645 2/20 0.48
HDAC8 Q9BY41 1/20 0.47
TNF P01375 1/20 0.47
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19846982 0.89 HTR2A (0.68) HTR2AGPR84SOS1KDM4ELMNA
SCHEMBL10078148 0.89 HTR2A (0.68) HTR2AGPR84SOS1KDM4ELMNA
SCHEMBL128685 0.88 KMT2A (0.66) HTR2AGPR84SOS1PTPRAKDM4E
SCHEMBL10958198 0.88 SCN9A (0.59) HTR2AGPR84SOS1PTPRAKDM4E
SCHEMBL623336 0.88 KMT2A (0.66) HTR2AGPR84SOS1PTPRAKDM4E
SCHEMBL456668 0.88 KMT2A (0.66) HTR2AGPR84SOS1PTPRAKDM4E
SCHEMBL18029175 0.88 KMT2A (0.66) HTR2AGPR84SOS1PTPRAKDM4E
SCHEMBL30381542 0.88 KMT2A (0.66) HTR2AGPR84SOS1PTPRAKDM4E
SCHEMBL29405769 0.88 KMT2A (0.66) HTR2AGPR84SOS1PTPRAKDM4E
SCHEMBL18427690 0.86 HTR2A (0.51) HTR2AGPR84SOS1PTPRAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180037917-A1 PROTECTING GROUP CHEMISTRY FOR CLEAN, REDUCTANT-FREE DYEING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-02-08 US disclosed
WO-2012173846-A2 PEPTIDOMIMETIC MACROCYCLES AILERON THERAPEUTICS, INC. (US) 2012-12-20 WO disclosed
WO-2012021875-A1 PEPTIDOMIMETIC MACROCYCLES WITH TRIAZOLE LINKERS AILERON THERAPEUTICS, INC. (US) 2012-02-16 WO disclosed