SCHEMBL10080284

SCHEMBL10080284

CCc1c(Oc2cccc(N3CCN(C)CC3)c2)ccnc1C(C)NS(=O)(=O)c1ccc(C)c(Cl)cccc(C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.38
BRD4 O60885 2/20 0.38
GUSB P08236 3/20 0.37
HTR2C P28335 3/20 0.36
HTR1A P08908 1/20 0.36
HTR2A P28223 1/20 0.36
HTR7 P34969 1/20 0.36
DRD3 P35462 1/20 0.36
HTR6 P50406 1/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CCR8 P51685 1/20 0.35
BCL2 P10415 1/20 0.35
EGFR P00533 3/20 0.35
ALK Q9UM73 1/20 0.35
NUAK1 O60285 1/20 0.35
NUAK2 Q9H093 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12156234 0.90 SMN1; SMN2 (0.40) SMN1; SMN2BRD4GUSBHTR2CHTR1A
SCHEMBL1706072 0.88 HTR6 (0.46) RAD52SMN1; SMN2BRD4GUSBHTR2C
SCHEMBL1706085 0.77 SMN1; SMN2 (0.40) SMN1; SMN2BRD4GUSBHTR2CHTR1A
SCHEMBL1705567 0.77 SMN1; SMN2 (0.40) SMN1; SMN2BRD4GUSBHTR2CHTR1A
SCHEMBL1705603 0.77 SMN1; SMN2 (0.40) SMN1; SMN2BRD4GUSBHTR2CHTR1A
SCHEMBL12156232 0.76 HTR6 (0.43) RAD52SMN1; SMN2BRD4GUSBHTR2C
SCHEMBL1705585 0.74 ADRA2C (0.41) HTR6MAPTMEN1KMT2AEGFR
SCHEMBL1706545 0.74 HRH4 (0.41) HTR6MAPTMEN1KMT2AEGFR
SCHEMBL12161117 0.74 S1PR1 (0.56) RAD52SMN1; SMN2BRD4GUSBHTR2C
SCHEMBL12156278 0.73 SMN1; SMN2 (0.39) SMN1; SMN2BRD4GUSBHTR2CHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2177512-B1 INHIBITOR OF BINDING OF S1P1 TAISHO PHARMACEUTICAL CO LTD (JP) 2012-04-18 EP disclosed