SCHEMBL10080360

SCHEMBL10080360

CN1CCN(c2ccc(Nc3nccc(-c4ccc(N5CCCC5)c(N)c4)n3)cn2)CC1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 9/20 0.57
CDK2 P24941 9/20 0.57
CCNA1 P78396 9/20 0.57
ZAP70 P43403 2/20 0.57
STK17A Q9UEE5 2/20 0.55
MYLK4 Q86YV6 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
TBK1 Q9UHD2 1/20 0.55
CDK4 P11802 3/20 0.53
CCND3 P30281 3/20 0.53
GSK3B P49841 3/20 0.53
PIM1 P11309 2/20 0.53
MTOR P42345 2/20 0.53
SMG1 Q96Q15 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL434273 0.87 TBK1 (0.61) CCNA2CDK2CCNA1ZAP70STK17A
SCHEMBL10081567 0.84 ZAP70 (0.50) CCNA2CDK2CCNA1ZAP70STK17A
SCHEMBL10080361 0.83 CCNA2 (0.47) CCNA2CDK2CCNA1ZAP70STK17A
SCHEMBL10080738 0.82 JAK2 (0.59) CCNA2CDK2CCNA1CDK4CCND3
SCHEMBL10081121 0.80 JAK2 (0.57) CCNA2CDK2CCNA1ZAP70STK17A
SCHEMBL29618397 0.78 CCNA2 (0.65) CCNA2CDK2CCNA1ZAP70CLK4
SCHEMBL29618396 0.78 CCNA2 (0.65) CCNA2CDK2CCNA1ZAP70CLK4
SCHEMBL15986738 0.78 ZAP70 (0.54) CCNA2CDK2CCNA1ZAP70STK17A
SCHEMBL10080355 0.76 TBK1 (0.59) CDK2ZAP70STK17AMYLK4CLK4
SCHEMBL13467178 0.76 TBK1 (0.52) ZAP70STK17AMYLK4CLK4TBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012010826-A1 PYRIMIDINE COMPOUNDS AS INHIBITORS OF PROTEIN KINASES IKK EPSILON AND/OR TBK-1, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DOMAINEX LIMITED (GB) 2012-01-26 WO disclosed