SCHEMBL1008207

SCHEMBL1008207

CC(=O)On1nc(C(F)(F)F)c2c1CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.38
ADORA1 P30542 2/20 0.38
NR1H2 P55055 1/20 0.37
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
PARP1 P09874 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
MAPT P10636 2/20 0.34
C5AR1 P21730 1/20 0.34
F12 P00748 2/20 0.34
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
HPGDS O60760 1/20 0.34
CTSS P25774 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1005208 0.91 ADORA1 (0.40) ESR2ADORA1NR1H2PARP1TNKS2
SCHEMBL4760408 0.83 DPP4 (0.47) ESR2ADORA1NR1H2DDB1CRBN
SCHEMBL18852439 0.81 ESR2 (0.39) ESR2ADORA1NR1H2DDB1CRBN
SCHEMBL4762470 0.80 DPP4 (0.49) ESR2ADORA1NR1H2HDAC1HDAC6
SCHEMBL1008205 0.79 LMNA (0.56) ADORA1DDB1CRBNCTSS
SCHEMBL15730073 0.76 DPP4 (0.47) ESR2ADORA1NR1H2PARP1TNKS2
SCHEMBL1007338 0.75 TRPM2 (0.45) ADORA1MAPT
SCHEMBL14555911 0.74 ADORA1 (0.41) ESR2ADORA1NR1H2DDB1CRBN
SCHEMBL15730211 0.74 DPP4 (0.38) ADORA1NR1H2DDB1CRBNDPP4
SCHEMBL17066905 0.74 ADORA1 (0.42) ESR2ADORA1NR1H2DPP4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2269990-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2011-01-05 EP disclosed