SCHEMBL1008750

SCHEMBL1008750

N#Cc1ncc(CC(N)=O)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
CA2 P00918 1/20 0.33
CPB2 Q96IY4 1/20 0.33
S100A9 P06702 1/20 0.33
TBK1 Q9UHD2 1/20 0.32
MAOB P27338 1/20 0.32
PRKAB2 O43741 1/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA2 P54646 1/20 0.32
PRKAA1 Q13131 1/20 0.32
PRKAG3 Q9UGI9 1/20 0.32
PRKAG2 Q9UGJ0 1/20 0.32
PRKAB1 Q9Y478 1/20 0.32
AR P10275 1/20 0.31
CYP11B2 P19099 1/20 0.31
ADRA1D P25100 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL335184 0.78 ALDH1A1 (0.41) TDP1KDM4EALDH1A1POLBS100A9
SCHEMBL1008889 0.76 POLB (0.42) TDP1KDM4EALDH1A1POLBS100A9
SCHEMBL15157663 0.76 ALDH1A1 (0.36) TDP1KDM4EALDH1A1POLBTBK1
SCHEMBL16879533 0.75 ALDH1A1 (0.41) KDM4EALDH1A1POLBS100A9HTT
SCHEMBL10314907 0.75 ALDH1A1 (0.41) TDP1KDM4EALDH1A1POLBS100A9
SCHEMBL1010296 0.75 KDM4E (0.41) TDP1KDM4EALDH1A1POLBS100A9
SCHEMBL1060088 0.72 ALDH1A1 (0.40) TDP1KDM4EALDH1A1POLBMAOB
SCHEMBL12499186 0.71 ADRA1D (0.51) KDM4EALDH1A1CA2ARADRA1D
SCHEMBL22561720 0.71 KDM4E (0.38) KDM4EALDH1A1POLB
SCHEMBL22713562 0.71 KDM4E (0.38) KDM4EALDH1A1POLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268618-A1 COMPOUNDS AND COMPOSITIONS AS TLR ACTIVITY MODULATORS IRM LLC (BM) 2011-01-05 EP disclosed
WO-2009111337-A1 COMPOUNDS AND COMPOSITIONS AS TLR ACTIVITY MODULATORS IRM LLC (BM) 2009-09-11 WO disclosed