SCHEMBL10100401

SCHEMBL10100401

CCCC=CNC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.40
CA7 P43166 2/20 0.40
CA12 O43570 2/20 0.40
CA14 Q9ULX7 2/20 0.40
CTSK P43235 13/20 0.38
TDP1 Q9NUW8 1/20 0.36
CA2 P00918 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CTSS P25774 1/20 0.35
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
MAPK10 P53779 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10776406 1.00 CA1 (0.40) CA1CA7CA12CA14CTSK
SCHEMBL28556471 0.86 CNR1 (0.44) TDP1KMT2AMEN1
SCHEMBL12492444 0.86 CNR1 (0.44) TDP1KMT2AMEN1
SCHEMBL571467 0.85 CTSK (0.40) CA1CA7CA12CA14CTSK
SCHEMBL20159624 0.85 CTSK (0.40) CA1CA7CA12CA14CTSK
SCHEMBL16061377 0.85 CTSK (0.40) CA1CA7CA12CA14CTSK
SCHEMBL6111877 0.82 CTSK (0.40) CA1CA7CA12CA14CTSK
SCHEMBL7442687 0.82 CA1 (0.40) CA1CA7CA12CA14CTSK
SCHEMBL7442690 0.82 CA1 (0.40) CA1CA7CA12CA14CTSK
SCHEMBL166206 0.81 CA1 (0.42) CA1CA7CA12CA14CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097750-B2 Highly enantioselective, converting aromatic and aliphatic aldehydes into optically active aryl and alkyl beta -amino acids BRANDEIS UNIVERSITY (US) 2012-01-17 US disclosed
US-20080228000-A1 Cinchona Alkaloid-Catalyzed Asymmetric Mannich Reactions BRANDEIS UNIVERSITY (US) 2008-09-18 US disclosed
EP-0229944-A2 Novel tetrahydroisoquinoline derivatives SYNTEX (U.S.A.) INC. (US) 1987-07-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080228000-A1 Cinchona Alkaloid-Catalyzed Asymmetric Mannich Reactions MANBA, MAN2A1, ASNS CA1 456/4885CA7 34/4885CA12 266/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.