SCHEMBL10104440

SCHEMBL10104440

COc1c(C)cc(C(C)(C)C)cc1CN1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 1/20 0.47
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CNR2 P34972 5/20 0.41
CNR1 P21554 2/20 0.40
SYK P43405 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10104443 0.87 ALDH1A1 (0.47) SMN1; SMN2KDM4EPOLBCYP3A4HTT
SCHEMBL5124007 0.86 SMN1; SMN2 (0.40) CYP2A13SMN1; SMN2CYP3A4CYP2D6CNR2
SCHEMBL10104438 0.86 ALDH1A1 (0.49) KDM4EPOLBCYP3A4CYP2D6HTT
SCHEMBL13130492 0.84 MAPT (0.45) CYP2A13SMN1; SMN2HTT
SCHEMBL14943431 0.84 TP53 (0.51) CYP2A13PKMSMN1; SMN2KDM4EPOLB
SCHEMBL10030806 0.83 SMN1; SMN2 (0.51) CYP2A13PKMSMN1; SMN2KDM4EPOLB
SCHEMBL5124004 0.81 HCRTR1 (0.42) SMN1; SMN2KDM4ECNR2CNR1HTT
SCHEMBL2621005 0.78 CYP2C9 (0.57) CYP2A13KDM4ECYP3A4CYP2D6HTT
SCHEMBL5114806 0.75 ALOX5AP (0.44) CYP2A13SMN1; SMN2KDM4EHTT
SCHEMBL12809477 0.75 SIGMAR1 (0.45) PKMSMN1; SMN2KDM4EPOLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8778929-B2 Substituted heteroaryl inhibitors of B-RAF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-07-15 US disclosed
US-8653087-B2 Pyrido [5, 4-D] pyrimidines as cell proliferation inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-02-18 US disclosed
US-20120094975-A1 PYRIDO [5, 4-D] PYRIMIDINES AS CELL PROLIFERATION INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-04-19 US disclosed
US-20110312939-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-12-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110312939-A1 NEW CHEMICAL COMPOUNDS CCNA1, CCNT1, MKI67 CYP2A13 370/4885PKM 1901/4885SMN1; SMN2 1280/4885
US-20120094975-A1 PYRIDO [5, 4-D] PYRIMIDINES AS CELL PROLIFERATION INHIBITORS CCNT1, CCNA1, CCND1 CYP2A13 1507/4885PKM 854/4885SMN1; SMN2 521/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.