SCHEMBL10104773

SCHEMBL10104773

C#CCn1c(=O)c2[nH]c(-c3cn(Cc4cccc(C)c4)nn3)nc2n(C)c1=O

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.51
ADORA2B P29275 17/20 0.51
ADORA1 P30542 17/20 0.51
ADORA3 P0DMS8 11/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9904021 0.89 ADORA2B (0.60) ADORA2AADORA2BADORA1ADORA3
SCHEMBL10104730 0.82 ADORA2B (0.60) ADORA2AADORA2BADORA1ADORA3
SCHEMBL9903991 0.76 ADORA2A (0.72) ADORA2AADORA2BADORA1ADORA3
SCHEMBL9904033 0.75 ADORA2B (0.75) ADORA2AADORA2BADORA1ADORA3
SCHEMBL8183967 0.72 ADORA1 (0.55) ADORA2AADORA2BADORA1
SCHEMBL10104740 0.71 MAOB (0.57)
SCHEMBL9904195 0.71 ADORA2B (0.73) ADORA2AADORA2BADORA1ADORA3
SCHEMBL9904089 0.69 ADORA2B (0.55) ADORA2AADORA2BADORA1ADORA3
SCHEMBL3949936 0.68 ADORA2B (0.59) ADORA2AADORA2BADORA1ADORA3
SCHEMBL1944369 0.67 ADORA2B (1.00) ADORA2AADORA2BADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465859-A1 8-Triazolylxanthine derivatives, processes for their production and their use as adenosine receptor antagonists Life & Brain GmbH (DE) 2012-06-20 EP disclosed