SCHEMBL10108494

SCHEMBL10108494

Cc1cccc(Cl)c1-c1cc2cnc(Nc3ccncc3)nc2n(C)c1=O

nearest known ligand 0.89

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 12/20 0.89
FGFR1 P11362 10/20 0.89
EGFR P00533 8/20 0.89
WEE1 P30291 6/20 0.85
PDGFRB P09619 8/20 0.75
PDGFRA P16234 8/20 0.75
ABL1 P00519 7/20 0.75
MAPK14 Q16539 7/20 0.75
FGFR2 P21802 1/20 0.74
FGFR4 P22455 1/20 0.74
FGFR3 P22607 1/20 0.74
KIT P10721 3/20 0.74
STAT5A P42229 1/20 0.69
ACVR1 Q04771 1/20 0.69
PKMYT1 Q99640 1/20 0.69
PSEN1 P49768 1/20 0.68
PSEN2 P49810 1/20 0.68
APH1B Q8WW43 1/20 0.68
NCSTN Q92542 1/20 0.68
APH1A Q96BI3 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL868353 0.94 FGFR1 (1.00) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL25779595 0.92 WEE1 (1.00) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL17520126 0.91 SRC (0.90) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL10108142 0.89 FGFR1 (0.87) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL5762046 0.86 SRC (1.00) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL1249524 0.86 FGFR1 (1.00) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL2083696 0.85 SRC (1.00) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL5763306 0.85 FGFR1 (1.00) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL5764062 0.85 FGFR1 (1.00) SRCFGFR1EGFRWEE1PDGFRB
SCHEMBL4747103 0.83 SRC (0.81) SRCFGFR1EGFRWEE1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120077811-A1 PRODRUG FORMS OF KINASE INHIBITORS AND THEIR USE IN THERAPY AUCKLAND UNISERVICES LIMITED (NZ) 2012-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120077811-A1 PRODRUG FORMS OF KINASE INHIBITORS AND THEIR USE IN THERAPY NTRK3, TK1, TNNI3K SRC 176/4885FGFR1 115/4885EGFR 48/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.