SCHEMBL10112852

SCHEMBL10112852

O=C(O)c1cccc(OCC2CCN(c3ccc([N+](=O)[O-])cn3)CC2)c1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 12/20 0.64
SOAT1 P35610 2/20 0.64
CYP3A4 P08684 1/20 0.64
SOAT2 O75908 1/20 0.51
DGAT2 Q96PD7 1/20 0.51
MAPT P10636 4/20 0.51
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ATM Q13315 1/20 0.48
NR1H4 Q96RI1 1/20 0.48
ALDH1A1 P00352 1/20 0.47
NPY2R P49146 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669645 0.90 DGAT1 (0.54) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL1444238 0.84 DGAT1 (0.68) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL670183 0.78 MAPT (0.48) DGAT1SOAT1CYP3A4MAPTPOLB
SCHEMBL10113679 0.78 DGAT1 (1.00) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113332 0.77 DGAT1 (0.86) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL5453369 0.77 L3MBTL1 (0.70) MAPTPOLBL3MBTL1MEN1KMT2A
SCHEMBL3542849 0.77 MAPT (0.64) MAPTKDM4EPOLBL3MBTL1MEN1
SCHEMBL3542851 0.77 MAPT (0.64) MAPTKDM4EPOLBL3MBTL1MEN1
SCHEMBL10112844 0.77 DGAT1 (0.81) DGAT1SOAT1CYP3A4SOAT2DGAT2
SCHEMBL10113345 0.77 DGAT1 (0.75) DGAT1SOAT1CYP3A4SOAT2DGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012024179-A1 SUBSTITUTED AMIDE DERIVATIVES AS DGAT-1 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-02-23 WO disclosed